SCHEMBL1637468

SCHEMBL1637468

CCCCCOC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@@H](O)[C@@H]1O

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EHMT1 Q9H9B1 1/20 0.76
RXFP1 Q9HBX9 1/20 0.69
ADORA1 P30542 3/20 0.65
SMN1; SMN2 Q16637 2/20 0.65
ADORA3 P0DMS8 2/20 0.65
ADORA2A P29274 2/20 0.65
ADORA2B P29275 2/20 0.65
DPP4 P27487 1/20 0.65
MEN1 O00255 1/20 0.65
SLC28A1 O00337 1/20 0.65
MAP3K7 O43318 1/20 0.65
SLC28A2 O43868 1/20 0.65
GAPDH P04406 1/20 0.65
MAPK1 P28482 1/20 0.65
STAT6 P42226 1/20 0.65
PI4KA P42356 1/20 0.65
KMT2A Q03164 1/20 0.65
PI4K2B Q8TCG2 1/20 0.65
DOT1L Q8TEK3 1/20 0.65
SLC29A1 Q99808 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9231760 1.00 EHMT1 (0.76) EHMT1RXFP1ADORA1SMN1; SMN2ADORA3
SCHEMBL10865966 0.99 EHMT1 (0.74) EHMT1RXFP1ADORA1SMN1; SMN2ADORA3
SCHEMBL1920531 0.99 EHMT1 (0.74) EHMT1RXFP1ADORA1SMN1; SMN2ADORA3
SCHEMBL8671037 0.97 EHMT1 (0.74) EHMT1RXFP1ADORA1SMN1; SMN2ADORA3
SCHEMBL8671033 0.97 EHMT1 (0.74) EHMT1RXFP1ADORA1SMN1; SMN2ADORA3
SCHEMBL29936475 0.97 EHMT1 (0.74) EHMT1RXFP1ADORA1SMN1; SMN2ADORA3
SCHEMBL5562010 0.94 EHMT1 (0.67) EHMT1RXFP1ADORA1SMN1; SMN2ADORA3
SCHEMBL2534140 0.93 EHMT1 (0.70) EHMT1RXFP1ADORA1SMN1; SMN2ADORA3
SCHEMBL10590849 0.91 EHMT1 (0.66) EHMT1RXFP1ADORA1SMN1; SMN2ADORA3
SCHEMBL8970443 0.91 EHMT1 (0.63) EHMT1RXFP1ADORA1SMN1; SMN2ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4069382-A 9-(5-O-Acyl-β-D-arabinofuranosyl)adenine compounds PARKE, DAVIS & COMPANY (US) 1978-01-17 US claimed
US-20110265195-A1 UNIQUE ASSOCIATED KAPOSI'S SARCOMA VIRUS SEQUENCES AND USES THEREOF THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2011-10-27 US disclosed
US-7932066-B2 Unique associated kaposi's sarcoma virus sequences and uses thereof THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2011-04-26 US disclosed
US-20090022748-A1 Unique associated Kaposi's sarcoma virus sequences and uses thereof CHANG YUAN 2009-01-22 US disclosed
US-6500663-B1 TREATING A SUBJECT AFFLICTED WITH A KAPOSI'S SARCOMA CAUSED BY KAPOSI'S SARCOMA ASSOCIATED HERPESVIRUS WHICH COMPRISES ADMINISTERING A NUCLEOSIDE ANALOG OR AN ANTISENSE NUCLEIC ACID THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2002-12-31 US disclosed
US-6348586-B1 NUCLEOTIDE SEQUENCE OF HERPES VIRUS; DIAGNOSIS; VACCINES; VIRICIDES; ANTISENSE AGENTS; TRIPLEX OLIGONUCLEOTIDES; THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2002-02-19 US disclosed
US-6183751-B1 VACCINES; DIAGNOSIS; OPEN READING FRAME; GENETIC ENGINEERING THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2001-02-06 US disclosed
US-6150093-A NUCLEOTIDE SEQUENCES PREFERENTIAL FOR HERPES VIRUS ASSOCIATED WITH A CANCER; FOR TREATMENT, DIAGNOSIS AND DETECTION OF AQUIRED IMMUNODEFICIENCY SYNDROME RELATED CANCER THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2000-11-21 US disclosed
US-6093550-A DIAGNOSING KAPOSI'S SARCOMA(KS) ASSOCIATED HERPESVIRUS INFECTION BY CONTACTING A SAMPLE WITH A KS ASSOCIATED HERPESVIRUS ANTIGEN, DETERMINING THE LEVEL OF KS ASSOCIATED HERPESVIRUS ANTIBODY BOUND TO THE ANTIGEN; IMMUNOASSAY KITS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2000-07-25 US disclosed
EP-0804547-A4 UNIQUE ASSOCIATED KAPOSI'S SARCOMA VIRUS SEQUENCES AND USES THEREOF UNIV COLUMBIA (US) 1999-11-03 EP disclosed
WO-1998004576-A1 UNIQUE ASSOCIATED KAPOSI'S SARCOMA VIRUS SEQUENCES AND USES THEREOF THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 1998-02-05 WO disclosed
EP-0804547-A1 UNIQUE ASSOCIATED KAPOSI'S SARCOMA VIRUS SEQUENCES AND USES THEREOF The Trustees of Columbia University in the City of New York (US) 1997-11-05 EP disclosed
WO-1997027208-A1 UNIQUE ASSOCIATED KAPOSI'S SARCOMA VIRUS SEQUENCES AND USES THEREOF THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 1997-07-31 WO disclosed
EP-0726708-A1 VIRUS ASSOCIATED MULTIPLE SCLEROSIS: TREATMENTS, PREVENTION AND DIAGNOSIS THEREOF PATHOGENESIS CORPORATION (US) 1996-08-21 EP disclosed
WO-1996015779-A1 UNIQUE ASSOCIATED KAPOSI'S SARCOMA VIRUS SEQUENCES AND USES THEREOF THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 1996-05-30 WO disclosed
WO-1996006159-A1 UNIQUE ASSOCIATED KAPOSI'S SARCOMA VIRUS SEQUENCES AND USES THEREOF THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 1996-02-29 WO disclosed
WO-1995012313-A1 VIRUS ASSOCIATED MULTIPLE SCLEROSIS: TREATMENTS, PREVENTION AND DIAGNOSIS THEREOF PATHOGENESIS CORPORATION (US) 1995-05-11 WO disclosed
EP-0317728-A2 Use of 9-(beta-D-arabinofuranosyl) adenine derivatives for the preparation of pharmaceutical compositions for the treatment of aids WARNER-LAMBERT COMPANY (US) 1989-05-31 EP disclosed
US-4069382-A 9-(5-O-Acyl-β-D-arabinofuranosyl)adenine compounds PARKE, DAVIS & COMPANY (US) 1978-01-17 US disclosed
US-4069382-A 9-(5-O-Acyl-β-D-arabinofuranosyl)adenine compounds PARKE, DAVIS & COMPANY (US) 1978-01-17 US disclosed