SCHEMBL16374698

SCHEMBL16374698

CC(C)(C)c1ccc(C(=O)Nc2cc(NCc3ccc(CF)cc3)n3nccc3n2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 10/20 0.48
KCNN3 Q9UGI6 3/20 0.42
KCNN1 Q92952 1/20 0.40
KCNN2 Q9H2S1 1/20 0.40
NAMPT P43490 1/20 0.40
MEN1 O00255 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C19 P33261 1/20 0.40
KMT2A Q03164 1/20 0.40
MAPKAPK2 P49137 1/20 0.40
CDK2 P24941 3/20 0.40
CCNE1 P24864 2/20 0.40
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
NFKB1 P19838 1/20 0.39
RAB9A P51151 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1523957 0.92 MAP3K5 (0.48) MAP3K5KCNN3KCNN1KCNN2NAMPT
SCHEMBL1072279 0.90 KCNN3 (0.52) MAP3K5KCNN3KCNN1KCNN2MAPKAPK2
SCHEMBL1019238 0.89 NPC1 (0.52) MAP3K5KCNN3MEN1KMT2ANPC1
SCHEMBL1523648 0.88 KCNN3 (0.48) MAP3K5KCNN3CDK2CCNE1NPC1
SCHEMBL1523690 0.87 CA2 (0.53) MAP3K5NAMPTMEN1KMT2A
SCHEMBL1016782 0.87 KCNN3 (0.47) MAP3K5KCNN3KCNN1KCNN2MAPKAPK2
SCHEMBL1523664 0.85 KCNN3 (0.57) MAP3K5KCNN3KCNN1KCNN2KMT2A
SCHEMBL1523277 0.85 CDK2 (0.57) MAP3K5NAMPTMEN1KMT2ACDK2
SCHEMBL1523231 0.84 TSHR (0.46) MAP3K5MEN1KMT2ANPC1MAPT
SCHEMBL12838103 0.84 MAP3K5 (0.46) MAP3K5KCNN3CDK2RETGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8921358-B2 Apoptosis signal-regulating kinase 1 inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2014-12-30 US disclosed