SCHEMBL163752

SCHEMBL163752

NCCc1ncc(-c2ccc(NC(=O)Nc3cc(F)c(F)cc3F)cc2)s1

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 8/20 0.58
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA9 Q16790 1/20 0.48
NTRK1 P04629 1/20 0.42
CNR1 P21554 1/20 0.40
KDR P35968 8/20 0.39
PDGFRB P09619 5/20 0.39
KIT P10721 2/20 0.38
FLT3 P36888 2/20 0.38
LCK P06239 1/20 0.38
CSF1R P07333 1/20 0.38
FLT1 P17948 1/20 0.38
FLT4 P35916 1/20 0.38
RIPK1 Q13546 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL163660 0.99 DGAT1 (0.57) DGAT1CA12CA1CA2CA9
SCHEMBL12503659 0.88 DGAT1 (0.53) DGAT1CA12CA1CA2CA9
SCHEMBL15021985 0.88 DGAT1 (0.59) DGAT1CA12CA1CA2CA9
SCHEMBL161687 0.87 DGAT1 (0.55) DGAT1NTRK1CNR1KDRKIT
Hydrochloric Acid SCHEMBL161482 0.86 DGAT1 (0.54) DGAT1NTRK1CNR1KDRKIT
SCHEMBL158731 0.85 DGAT1 (0.54) DGAT1CA12CA1CA2CA9
SCHEMBL159242 0.83 DGAT1 (0.51) DGAT1CA12CA1CA2CA9
SCHEMBL15022135 0.83 DGAT1 (0.53) DGAT1CA12CA1CA2CA9
SCHEMBL15022044 0.81 DGAT1 (0.52) DGAT1CA12CA1CA2CA9
Hydrochloric Acid SCHEMBL160270 0.81 DGAT1 (0.57) DGAT1CNR1KDRKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611783-A2 HETEROCYCLIC COMPOUNDS AS DGAT1 INHIBITORS Piramal Enterprises Limited (IN) 2013-07-10 EP disclosed
WO-2012029032-A2 HETEROCYCLIC COMPOUNDS AS DGAT1 INHIBITORS PIRAMAL LIFE SCIENCES LIMITED (IN) 2012-03-08 WO disclosed