SCHEMBL16375362

SCHEMBL16375362

c1ccc(CNc2ncnc3sc(-c4ccccc4)cc23)cc1

nearest known ligand 0.82

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EGFR P00533 7/20 0.82
KDM4E B2RXH2 3/20 0.67
ALDH1A1 P00352 3/20 0.67
LMNA P02545 1/20 0.67
RCE1 Q9Y256 1/20 0.67
MEN1 O00255 3/20 0.67
KMT2A Q03164 3/20 0.67
ICAM1 P05362 1/20 0.67
SELE P16581 1/20 0.67
VCAM1 P19320 1/20 0.67
POLB P06746 1/20 0.66
RAD52 P43351 1/20 0.66
HPGD P15428 1/20 0.62
FGFR1 P11362 3/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16375364 0.84 EGFR (0.71) EGFRKDM4EALDH1A1LMNARCE1
SCHEMBL29360504 0.82 ICAM1 (0.72) EGFRKDM4ELMNAICAM1SELE
SCHEMBL4800479 0.82 TEK (0.66) EGFRKDM4EALDH1A1LMNARCE1
SCHEMBL4803681 0.81 EGFR (0.58) EGFRKDM4EALDH1A1LMNARCE1
SCHEMBL17200798 0.81 FDPS (0.78) EGFRKDM4EALDH1A1LMNARCE1
SCHEMBL5429540 0.80 ICAM1 (1.00) EGFRKDM4EALDH1A1LMNAMEN1
SCHEMBL15503823 0.80 RAD52 (1.00) EGFRKDM4EALDH1A1LMNARCE1
SCHEMBL11414153 0.77 EGFR (0.64) EGFRLMNAICAM1SELEVCAM1
SCHEMBL16376062 0.76 EGFR (1.00) EGFRICAM1SELEVCAM1
SCHEMBL16375358 0.74 EGFR (1.00) EGFRICAM1SELEVCAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015000959-A1 4-AMINO-6-ARYL[2,3-D]PYRIMIDINES FOR THE INHIBITION OF EGFR TYROSINE KINASE NORWEGIAN UNIVERSITY OF SCIENCE AND TECHNOLOGY (NTNU) (NO) 2015-01-08 WO disclosed