SCHEMBL16379337

SCHEMBL16379337

COC(=O)[C@H](C)COc1ccc(C(F)(F)F)cc1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.50
MAOB P27338 2/20 0.47
NOS3 P29474 2/20 0.44
NOS1 P29475 2/20 0.44
NOS2 P35228 2/20 0.44
PPARA Q07869 1/20 0.44
PPARD Q03181 3/20 0.44
PSMB5 P28074 1/20 0.44
MDH1 P40925 1/20 0.43
MDH2 P40926 1/20 0.43
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21991581 0.85 ALDH1A1 (0.48) ALDH1A1MAOBNOS3NOS1NOS2
SCHEMBL16379339 0.84 PPARA (0.49) ALDH1A1MAOBPPARAPPARDPSMB5
SCHEMBL22651641 0.82 ALDH1A1 (0.51) ALDH1A1
SCHEMBL17601685 0.82 S1PR1 (0.53) MAOBPPARA
SCHEMBL16915059 0.82 MAOB (0.44) MAOBNOS3NOS1NOS2PPARA
SCHEMBL17601686 0.82 S1PR1 (0.53) MAOBPPARA
SCHEMBL21992729 0.82 ALDH1A1 (0.45) ALDH1A1MAOBNOS3NOS1NOS2
SCHEMBL7749771 0.80 MAPT (0.51) ALDH1A1MAOB
SCHEMBL12384285 0.79 MTNR1A (0.58) LMNA
SCHEMBL21991978 0.79 MAOB (0.57) MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8933018-B2 Boron containing polybasic bacterial efflux pump inhibitors and therapeutic uses thereof REMPEX PHARMACEUTICALS, INC. (US) 2015-01-13 US disclosed