SCHEMBL1638258

SCHEMBL1638258

COC(=O)c1ccc(CN(Cc2ncc[nH]2)C(C)c2ncc[nH]2)cc1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
KDM4E B2RXH2 2/20 0.49
CXCR4 P61073 2/20 0.40
LOXL2 Q9Y4K0 1/20 0.37
MLYCD O95822 1/20 0.37
HSP90AA1 P07900 1/20 0.37
TAAR1 Q96RJ0 2/20 0.37
PKM P14618 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.35
FPR2 P25090 1/20 0.35
GAA P10253 1/20 0.35
HTT P42858 1/20 0.35
CYP4A11 Q02928 1/20 0.35
CYP2D6 P10635 1/20 0.35
TSHR P16473 1/20 0.35
AR P10275 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1637370 0.80 TAAR1 (0.40) ALDH1A1CXCR4TAAR1SMN1; SMN2CYP2D6
SCHEMBL1205909 0.80 CXCR4 (0.44) CXCR4FPR2
SCHEMBL1638559 0.80 CXCR4 (0.48) CXCR4TAAR1FPR2
SCHEMBL3742746 0.78 TAAR1 (0.39) ALDH1A1KDM4ECXCR4TAAR1PKM
SCHEMBL1638097 0.78 CXCR4 (0.47) CXCR4TAAR1
SCHEMBL1205352 0.78 CXCR4 (0.55) CXCR4
SCHEMBL1638648 0.78 KDM4E (0.46) ALDH1A1KDM4ELOXL2MLYCDHSP90AA1
SCHEMBL1206794 0.78 CXCR4 (0.54) CXCR4
SCHEMBL1292672 0.76 CXCR4 (0.49) CXCR4TAAR1SMN1; SMN2CYP2D6TSHR
SCHEMBL1204925 0.76 CXCR4 (0.41) CXCR4TAAR1SMN1; SMN2CYP2D6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110172212-A1 AMINE-BASED COMPOUND AND USE THEREOF KUREHA CORPORATION (JP) 2011-07-14 US disclosed
US-7932281-B2 Amine-based compound and use thereof KUREHA CORPORATION (JP) 2011-04-26 US disclosed
US-20070208007-A1 Amine-Based Compound and Use Thereof KUREHA CORPORATION (JP) 2007-09-06 US disclosed
EP-1724263-A1 BASIC AMINE COMPOUND AND USE THEREOF Kureha Corporation (JP) 2006-11-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110172212-A1 AMINE-BASED COMPOUND AND USE THEREOF NR0B2, NR5A2, NR1D2 ALDH1A1 2045/4885KDM4E 2406/4885CXCR4 86/4885
US-20070208007-A1 Amine-Based Compound and Use Thereof NR0B2, NR5A2, NR2E1 ALDH1A1 1901/4885KDM4E 2871/4885CXCR4 100/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.