SCHEMBL16396237

SCHEMBL16396237

COC(=O)c1cc2c(s1)CCN(C(=O)OC(C)(C)C)C2.COC(=O)c1cc2c(s1)CCNC2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 4/20 0.50
PNMT P11086 2/20 0.49
ESR2 Q92731 1/20 0.44
TPSAB1 Q15661 1/20 0.44
TPSD1 Q9BZJ3 1/20 0.44
TPSG1 Q9NRR2 1/20 0.44
NR1H2 P55055 2/20 0.43
BRD4 O60885 1/20 0.43
CREBBP Q92793 1/20 0.43
MAPK1 P28482 2/20 0.41
KDM4E B2RXH2 2/20 0.40
NPC1 O15118 1/20 0.40
HPGD P15428 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ADORA1 P30542 2/20 0.39
MAPT P10636 1/20 0.39
ITGB3 P05106 1/20 0.38
ITGA2B P08514 1/20 0.38
F10 P00742 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL978284 0.90 HDAC6 (0.59) HDAC6ESR2NR1H2BRD4CREBBP
SCHEMBL743782 0.82 HDAC6 (0.54) HDAC6ESR2TPSAB1TPSD1TPSG1
SCHEMBL7795097 0.82 HDAC6 (0.51) HDAC6ESR2NR1H2MAPK1KDM4E
SCHEMBL977061 0.82 PNMT (0.70) PNMTTPSAB1TPSD1TPSG1MAPK1
SCHEMBL27081538 0.81 HDAC6 (0.59) HDAC6ESR2NR1H2MAPK1KDM4E
SCHEMBL29964789 0.81 HDAC6 (0.61) HDAC6TPSAB1TPSD1TPSG1MAPK1
Hydrochloric Acid SCHEMBL6421343 0.81 PNMT (0.68) PNMTTPSAB1TPSD1TPSG1MAPK1
SCHEMBL1174513 0.80 HDAC6 (0.72) HDAC6ESR2NR1H2BRD4CREBBP
SCHEMBL8555269 0.80 HDAC6 (0.54) HDAC6PNMTESR2TPSAB1TPSD1
SCHEMBL6421478 0.79 NR1H2 (0.54) HDAC6PNMTESR2TPSAB1TPSD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3004057-A1 HETEROCYCLIC DERIVATIVES AND USE THEREOF C&C Research Laboratories (KR) 2016-04-13 EP disclosed
WO-2014196793-A1 HETEROCYCLIC DERIVATIVES AND USE THEREOF C&C RESEARCH LABORATORIES (KR) 2014-12-11 WO disclosed