SCHEMBL16398763

SCHEMBL16398763

CCOC(=O)C(=O)NNC(=O)c1ccccc1C(F)(F)F

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GAA P10253 7/20 0.51
LMNA P02545 2/20 0.51
KCNK3 O14649 2/20 0.49
KCNK9 Q9NPC2 2/20 0.49
F2R P25116 1/20 0.45
KDM4E B2RXH2 2/20 0.45
TDP1 Q9NUW8 2/20 0.45
ALDH1A1 P00352 2/20 0.44
HPGD P15428 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
HTT P42858 1/20 0.43
EPHX2 P34913 2/20 0.43
TSHR P16473 2/20 0.41
PTGES O14684 1/20 0.41
PTGS1 P23219 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25392 0.81 SCD (0.47) LMNAALDH1A1
SCHEMBL9830646 0.81 GAA (0.75) GAALMNAKCNK3KCNK9F2R
SCHEMBL5837400 0.80 TSHR (0.49) GAALMNAKCNK3KCNK9F2R
SCHEMBL28191716 0.79 RXFP1 (0.50) GAALMNAKCNK3KCNK9F2R
SCHEMBL6449862 0.78 GAA (0.62) GAALMNAKCNK3KCNK9KDM4E
SCHEMBL29775613 0.78 LMNA (0.46) GAALMNAKCNK3KCNK9F2R
SCHEMBL1738337 0.78 LMNA (0.46) GAALMNAKCNK3KCNK9F2R
SCHEMBL1994129 0.76 TSHR (0.67) GAALMNAKCNK3KCNK9KDM4E
SCHEMBL16399046 0.76 NPSR1 (0.53) GAAKDM4ETDP1ALDH1A1SMN1; SMN2
SCHEMBL20827130 0.76 GPR35 (0.60) GAAKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3022199-A1 CYANOTRIAZOLE COMPOUNDS Otsuka Pharmaceutical Co., Ltd. (JP) 2016-05-25 EP disclosed
WO-2015008872-A1 CYANOTRIAZOLE COMPOUNDS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2015-01-22 WO disclosed