SCHEMBL1640360

SCHEMBL1640360

CN(Cc1ccccc1)C(=O)c1cn(Cc2ccccc2)c(=O)cc1O

nearest known ligand 0.60

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 6/20 0.60
KMT2A Q03164 3/20 0.50
HPGD P15428 2/20 0.49
MEN1 O00255 2/20 0.48
ALDH1A1 P00352 1/20 0.48
HSP90AB1 P08238 1/20 0.46
HSD17B2 P37059 1/20 0.44
MAPT P10636 1/20 0.43
USP19 O94966 1/20 0.43
GAA P10253 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1640352 0.81 LMNA (0.55) KMT2AMEN1ALDH1A1MAPT
SCHEMBL1640573 0.78 BRD4 (0.65) HPGDALDH1A1MAPTGAA
SCHEMBL1641959 0.78 KDM4E (0.48) HSP90AA1KMT2AHPGDALDH1A1HSP90AB1
SCHEMBL1641929 0.76 CRHBP (0.61) ALDH1A1
SCHEMBL1641827 0.75 BRD4 (0.57) KMT2AMEN1MAPT
SCHEMBL20677835 0.75 HSP90AA1 (1.00) HSP90AA1KMT2AHPGDMEN1ALDH1A1
SCHEMBL1642053 0.74 MAPT (0.59) KMT2AHPGDMEN1ALDH1A1MAPT
SCHEMBL1640326 0.74 HSP90AA1 (0.58) HSP90AA1KMT2AHPGDMEN1ALDH1A1
SCHEMBL1642389 0.74 EGLN1 (0.48) ALDH1A1GAA
SCHEMBL1641629 0.72 BRD4 (0.59) KMT2AHPGDMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110098324-A1 PROLYL HYDROXYLASE INHIBITORS GLAXOSMITHKLINE LLC 2011-04-28 US disclosed
EP-2306828-A1 PROLYL HYDROXYLASE INHIBITORS Glaxosmithkline LLC (US) 2011-04-13 EP disclosed
WO-2009158315-A1 PROLYL HYDROXYLASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2009-12-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110098324-A1 PROLYL HYDROXYLASE INHIBITORS HIF1AN, EGLN2, EGLN3 HSP90AA1 789/4885KMT2A 759/4885HPGD 31/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.