SCHEMBL16411005

SCHEMBL16411005

NCc1ccc(OF)c(Cl)c1

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CSNK2A1 P68400 10/20 0.61
MRGPRX4 Q96LA9 1/20 0.46
ROCK2 O75116 2/20 0.42
ROCK1 Q13464 2/20 0.42
GLA P06280 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
PNMT P11086 2/20 0.41
CSNK2A2 P19784 1/20 0.40
CSNK2B P67870 1/20 0.40
CSNK2A3 Q8NEV1 1/20 0.40
TAAR1 Q96RJ0 1/20 0.39
PRKCA P17252 1/20 0.39
AKT1 P31749 1/20 0.39
RPS6KA1 Q15418 1/20 0.39
IDO1 P14902 2/20 0.38
LOX P28300 1/20 0.38
LOXL3 P58215 1/20 0.38
LOXL2 Q9Y4K0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL506373 0.80 CSNK2A1 (0.66) CSNK2A1MRGPRX4GLASMN1; SMN2TAAR1
SCHEMBL28467993 0.79 CSNK2A1 (0.60) CSNK2A1MRGPRX4ROCK2ROCK1GLA
SCHEMBL3118077 0.79 CSNK2A1 (0.56) CSNK2A1MRGPRX4ROCK2ROCK1
Hydrochloric Acid SCHEMBL856874 0.78 CSNK2A1 (0.67) CSNK2A1MRGPRX4GLASMN1; SMN2TAAR1
SCHEMBL506790 0.77 CSNK2A1 (0.75) CSNK2A1MRGPRX4GLASMN1; SMN2CSNK2A2
SCHEMBL4550411 0.77 CSNK2A1 (0.59) CSNK2A1MRGPRX4ROCK2ROCK1GLA
Hydrochloric Acid SCHEMBL3110229 0.76 CSNK2A1 (0.76) CSNK2A1MRGPRX4GLASMN1; SMN2CSNK2A2
SCHEMBL6215544 0.76 CSNK2A1 (1.00) CSNK2A1MRGPRX4ROCK2ROCK1GLA
Hydrochloric Acid SCHEMBL2716247 0.75 CSNK2A1 (0.60) CSNK2A1MRGPRX4GLASMN1; SMN2
Hydrochloric Acid SCHEMBL15350295 0.75 CSNK2A1 (0.60) CSNK2A1MRGPRX4GLASMN1; SMN2IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015009930-A2 NOVEL PHOSPHODIESTERASE INHIBITORS AND USES THEREOF THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2015-01-22 WO disclosed