SCHEMBL16416992

SCHEMBL16416992

O=C(c1ccc(-c2ccc3cc[nH]c3n2)cc1)N1CCCCC1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.56
GHSR Q92847 2/20 0.52
HPGD P15428 8/20 0.51
ALDH1A1 P00352 2/20 0.51
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
PKM P14618 1/20 0.50
MAPK1 P28482 1/20 0.48
RIPK1 Q13546 2/20 0.47
BRD4 O60885 1/20 0.46
TRPV3 Q8NET8 1/20 0.45
TSHR P16473 1/20 0.45
HDAC4 P56524 1/20 0.44
ATR Q13535 1/20 0.44
FASN P49327 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL857503 0.76 RIPK1 (0.64) GHSRHPGDMAPK1RIPK1
SCHEMBL16417008 0.74 HRH3 (0.53) PARP1ALDH1A1
SCHEMBL1355458 0.74 GHSR (0.71) GHSRHPGDALDH1A1NPC1RAB9A
SCHEMBL29944074 0.74 GHSR (0.71) GHSRHPGDALDH1A1NPC1RAB9A
SCHEMBL857458 0.72 IKBKB (0.63) HPGDALDH1A1RIPK1BRD4
SCHEMBL23675226 0.72 PLK4 (0.56) HPGDALDH1A1RIPK1
SCHEMBL16416385 0.72 PARP1 (1.00) PARP1HPGDALDH1A1NPC1RAB9A
SCHEMBL7132525 0.72 HPGD (1.00) HPGDALDH1A1MAPK1TSHR
SCHEMBL27479149 0.72 HPGD (1.00) HPGDALDH1A1MAPK1TSHR
SCHEMBL857035 0.71 IKBKB (0.64) RIPK1BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015011008-A1 7-AZAINDOLE DERIVATIVES AS PARP INHIBITORS SIGMA-TAU INDUSTRIE FARMACEUTICHE RIUNITE S.P.A. (IT) 2015-01-29 WO disclosed