SCHEMBL16448787

SCHEMBL16448787

C[C@@H]1COc2cc(O)ccc21

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.48
MAOA P21397 1/20 0.48
MAOB P27338 1/20 0.48
TMEM97 Q5BJF2 2/20 0.44
MGAM O43451 1/20 0.44
PTPN1 P18031 1/20 0.44
ESR1 P03372 1/20 0.44
ESR2 Q92731 1/20 0.44
TTR P02766 1/20 0.44
HTR2B P41595 1/20 0.43
SIGMAR1 Q99720 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8584200 1.00 CYP3A4 (0.48) CYP3A4MAOAMAOBTMEM97MGAM
SCHEMBL16649032 0.85 DRD3 (0.49) CYP3A4ESR1ESR2TTR
SCHEMBL9749181 0.81 CYP3A4 (0.46) CYP3A4MAOAMAOBTMEM97MGAM
SCHEMBL4347592 0.78 CA2 (0.53) CYP3A4MAOAMAOBTMEM97PTPN1
SCHEMBL21284826 0.78 CYP3A4 (0.49) CYP3A4MAOAMAOBTMEM97ESR1
SCHEMBL21284745 0.78 CA2 (0.53) CYP3A4MAOAMAOBTMEM97PTPN1
SCHEMBL6327487 0.78 TOP2A (0.42)
SCHEMBL30456628 0.78 TOP2A (0.42)
SCHEMBL21933120 0.78 TOP2A (0.42)
Catechol SCHEMBL28905345 0.78 DRD3 (0.47) CYP3A4MAOAMAOBESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8952185-B2 Production method of optically active dihydrobenzofuran derivative TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2015-02-10 US disclosed