SCHEMBL1645202

SCHEMBL1645202

CC(C)=CCn1ncc(-c2ccncc2)c1-c1c(F)cccc1F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.44
PTGS2 P35354 2/20 0.44
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
LMNA P02545 1/20 0.35
S1PR1 P21453 2/20 0.34
GCK P35557 1/20 0.33
ADORA3 P0DMS8 2/20 0.32
ADORA2A P29274 2/20 0.32
ADORA2B P29275 2/20 0.32
ADORA1 P30542 2/20 0.32
AKR1C3 P42330 1/20 0.32
AKR1C2 P52895 1/20 0.32
KMT2A Q03164 1/20 0.31
KDR P35968 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
NFKB1 P19838 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1648133 0.79 S1PR1 (0.40) PTGS1PTGS2NPC1RAB9ALMNA
SCHEMBL1646195 0.79 S1PR1 (0.52) NPC1RAB9ALMNAS1PR1AKR1C3
SCHEMBL1648437 0.75 MAPK13 (0.38) NPC1RAB9ALMNACSNK1DCSNK1E
SCHEMBL1554460 0.71 NPC1 (0.39) NPC1RAB9ALMNAS1PR1GCK
SCHEMBL1645859 0.71 CHRM1 (0.47) LMNAKMT2ASMN1; SMN2
SCHEMBL1646948 0.70 RIPK3 (0.36) NPC1RAB9ALMNAS1PR1AKR1C3
SCHEMBL1647081 0.68 S1PR1 (0.50) PTGS1PTGS2NPC1RAB9ALMNA
SCHEMBL1646288 0.68 S1PR1 (0.47) PTGS1PTGS2NPC1RAB9ALMNA
SCHEMBL6076416 0.63 MAPK14 (0.51) NPC1RAB9AS1PR1KDRALDH1A1
SCHEMBL2649168 0.63 LMNA (0.58) NPC1RAB9ALMNAKMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2784070-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2784073-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2784071-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2784072-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2308866-A1 Phenylpyri(mi)dinylpyrazoles and their use as fungicides Bayer CropScience AG (DE) 2011-04-13 EP disclosed