Bicarbonate

Bicarbonate

SCHEMBL16457191

CC(CCCC1CC1)NC(=O)C(c1ccc(CN2N=C(c3ccccc3)OCC2=O)cc1)C1CCCC1.O=C(O)O

nearest known ligand 0.34

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.34
MAPK14 Q16539 2/20 0.34
PTGES O14684 2/20 0.34
MAPK11 Q15759 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
TP53 P04637 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
TSHR P16473 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
C3AR1 Q16581 3/20 0.33
MCHR1 Q99705 2/20 0.33
HTR1E P28566 2/20 0.32
S1PR3 Q99500 2/20 0.32
MEN1 O00255 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
CHRM4 P08173 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL517645 0.90 PTGES (0.39) PTGESSMN1; SMN2C3AR1
SCHEMBL517327 0.90 PTGES (0.39) PTGESSMN1; SMN2C3AR1
SCHEMBL517193 0.88 PTGES (0.33) PTGESSMN1; SMN2TP53CYP1A2CYP3A4
SCHEMBL517153 0.87 PTGES (0.33) PTGESSMN1; SMN2C3AR1MEN1KMT2A
SCHEMBL10176573 0.87 PTGES (0.33) PTGESSMN1; SMN2C3AR1MEN1KMT2A
SCHEMBL517807 0.86 PTGES (0.31) PTGESSMN1; SMN2TP53CYP1A2CYP3A4
SCHEMBL517806 0.85 P4HB (0.32) PTGES
Bicarbonate SCHEMBL3693977 0.83 C3AR1 (0.45) CYP3A4TSHRC3AR1KMT2ACYP2C19
SCHEMBL3693796 0.82 C3AR1 (0.42) PTGESC3AR1KMT2A
SCHEMBL1194091 0.82 C3AR1 (0.42) PTGESC3AR1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2406215-B1 OXO-HETEROCYCLICALLY SUBSTITUTED ALKYL CARBOXYLIC ACIDS AND USE THEREOF BAYER IP GMBH (DE) 2014-04-16 EP disclosed