SCHEMBL16458337

SCHEMBL16458337

CCC(C(=O)O)c1cnc(-c2nn(Cc3ccccc3F)c3ncccc23)nc1N

nearest known ligand 0.63

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.61
KCNH2 Q12809 1/20 0.61
PDE5A O76074 8/20 0.55
GUCY1A1 Q02108 10/20 0.54
GUCY1B1 Q02153 10/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15519039 0.90 PDE5A (0.56) ADORA3KCNH2PDE5AGUCY1A1GUCY1B1
SCHEMBL327099 0.90 PDE5A (0.55) ADORA3KCNH2PDE5A
SCHEMBL7835258 0.86 ADORA3 (0.65) ADORA3KCNH2PDE5AGUCY1A1GUCY1B1
SCHEMBL16459108 0.85 PDE5A (0.51) ADORA3KCNH2PDE5AGUCY1A1GUCY1B1
SCHEMBL6222114 0.85 ADORA3 (0.57) ADORA3KCNH2PDE5AGUCY1A1GUCY1B1
SCHEMBL175343 0.85 ADORA3 (0.63) ADORA3KCNH2PDE5AGUCY1A1GUCY1B1
SCHEMBL16244821 0.85 ADORA3 (0.63) ADORA3KCNH2PDE5AGUCY1A1GUCY1B1
SCHEMBL15518999 0.84 PDE5A (0.49) ADORA3KCNH2PDE5AGUCY1A1GUCY1B1
SCHEMBL174830 0.83 ADORA3 (0.63) ADORA3KCNH2PDE5AGUCY1A1GUCY1B1
SCHEMBL15732812 0.83 ADORA3 (0.64) ADORA3KCNH2PDE5AGUCY1A1GUCY1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2682394-A1 1H-pyrazolo[3,4-b]pyridin-triazine derivatives and their use for the treatment or the prevention of cardiovascular diseases Bayer Intellectual Property GmbH (DE) 2014-01-08 EP disclosed