SCHEMBL16463166

SCHEMBL16463166

O=c1ccn(-c2ccccc2-c2ccc(F)cc2)c2ccccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 1/20 0.41
MAPK14 Q16539 2/20 0.39
ALDH1A1 P00352 2/20 0.38
ATM Q13315 1/20 0.36
GRM2 Q14416 2/20 0.36
CDC25A P30304 1/20 0.36
CDC25C P30307 1/20 0.36
PTGS2 P35354 2/20 0.36
NR4A2 P43354 1/20 0.36
PTGS1 P23219 1/20 0.36
GABRP O00591 1/20 0.35
GABRD O14764 1/20 0.35
TNKS O95271 1/20 0.35
PARP1 P09874 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRB1 P18505 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16462146 0.87 BRD4 (0.36) ALDH1A1ATM
SCHEMBL16464134 0.85 L3MBTL1 (0.40) ALDH1A1TNKSTNKS2
SCHEMBL16464113 0.82 NR1I2 (0.43) MAPK14ALDH1A1ATMGRM2
SCHEMBL16460867 0.82 ATM (0.40) MAPK14ATM
SCHEMBL16461217 0.81 POLB (0.40) ALDH1A1ATMTNKS2
SCHEMBL16461892 0.79 MAPT (0.42) ALDH1A1
SCHEMBL339069 0.79 KDM4E (0.44) ALDH1A1PTGS2PTGS1
SCHEMBL16463954 0.77 KDM4E (0.58) ALDH1A1PTGS2TNKSPARP1TNKS2
SCHEMBL16462273 0.74 MAPK14 (0.37) MAPK14
SCHEMBL16463034 0.74 ADRA2C (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8629162-B2 Modulators of ATP-binding cassette transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-01-14 US disclosed