SCHEMBL16465321

SCHEMBL16465321

NC(=O)c1c(N)nc(F)nc1-c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.45
GAA P10253 2/20 0.45
MEN1 O00255 2/20 0.45
PLAU P00749 2/20 0.42
POLB P06746 2/20 0.42
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 3/20 0.42
DHODH Q02127 2/20 0.42
CDC7 O00311 1/20 0.41
CCNE1 P24864 1/20 0.41
CDK2 P24941 1/20 0.41
DBF4 Q9UBU7 1/20 0.41
CYP1A2 P05177 1/20 0.41
MAP2K3 P46734 1/20 0.41
SRC P12931 1/20 0.40
BRAF P15056 1/20 0.40
KDR P35968 1/20 0.40
IKBKB O14920 1/20 0.40
XDH P47989 1/20 0.40
CSNK1A1 P48729 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16465331 0.77 GAA (0.45) KMT2AGAAMEN1POLBKDM4E
SCHEMBL4559594 0.77 CXCL12 (0.44) KMT2AGAAMEN1PLAUPOLB
SCHEMBL13826194 0.76 PDPK1 (0.37) KMT2AMEN1POLBKDM4EALDH1A1
SCHEMBL18351964 0.76 DHODH (0.43) KMT2AGAAMEN1KDM4EDHODH
SCHEMBL15621840 0.76 CYP1A2 (0.51) KMT2AGAAMEN1PLAUPOLB
SCHEMBL15621964 0.73 NPC1 (0.50) KMT2AGAAMEN1IKBKBSMN1; SMN2
SCHEMBL15069721 0.71 KDR (0.64) KMT2AGAAMEN1POLBKDM4E
SCHEMBL1612494 0.71 IKBKB (0.48) KMT2AGAAMEN1POLBKDM4E
SCHEMBL14917472 0.70 CDC7 (0.45) KMT2AGAAMEN1POLBKDM4E
SCHEMBL14917475 0.70 IKBKB (0.51) KMT2AGAAMEN1PLAUKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2903970-A2 SUBSTITUTED PYRIMIDINYL KINASE INHIBITORS Portola Pharmaceuticals, Inc. (US) 2015-08-12 EP claimed
WO-2014058921-A2 SUBSTITUTED PYRIMIDINYL KINASE INHIBITORS PORTOLA PHARMACEUTICALS, INC. (US) 2014-04-17 WO claimed