SCHEMBL1646833

SCHEMBL1646833

CC(C)(C(=O)OCCBr)c1ccc([N+](=O)[O-])cc1.[O-][S+](Cl)Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
POLB P06746 1/20 0.44
GSK3B P49841 1/20 0.41
MAPT P10636 4/20 0.39
L3MBTL1 Q9Y468 2/20 0.38
ATM Q13315 1/20 0.38
RECQL P46063 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
CRHBP P24387 1/20 0.37
CRHR2 Q13324 1/20 0.37
ADRB2 P07550 1/20 0.36
ADRB1 P08588 1/20 0.36
ADRB3 P13945 1/20 0.36
GAA P10253 1/20 0.36
KDM4E B2RXH2 1/20 0.36
CYP2C19 P33261 1/20 0.36
CNR2 P34972 1/20 0.35
HSD11B1 P28845 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2231525 0.94 ALDH1A1 (0.49) ALDH1A1POLBGSK3BMAPTL3MBTL1
SCHEMBL1645876 0.79 PTPRC (0.48) ALDH1A1POLBMAPTL3MBTL1MEN1
SCHEMBL395369 0.78 ALDH1A1 (0.56) ALDH1A1POLBMAPTL3MBTL1KMT2A
SCHEMBL5491859 0.75 ALDH1A1 (0.52) ALDH1A1POLBMAPTL3MBTL1KMT2A
SCHEMBL429356 0.73 ALDH1A1 (0.65) ALDH1A1POLBMAPTL3MBTL1RECQL
SCHEMBL28359072 0.72 ALDH1A1 (0.51) ALDH1A1POLBMAPTGAAKDM4E
SCHEMBL2230940 0.72 GSK3B (0.53) ALDH1A1POLBGSK3BMAPTMEN1
SCHEMBL27030782 0.70 ALDH1A1 (0.53) ALDH1A1POLBMAPTMEN1KMT2A
SCHEMBL7221510 0.69 ATM (0.65) ALDH1A1POLBGSK3BMAPTL3MBTL1
SCHEMBL17055329 0.69 ALDH1A1 (0.55) ALDH1A1POLBMAPTL3MBTL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2303329-A1 ANTIFUNGAL COMBINATION THERAPY F2G Limited (GB) 2011-04-06 EP disclosed
WO-2009144473-A1 ANTIFUNGAL COMBINATION THERAPY F2G LIMITED (GB) 2009-12-03 WO disclosed