SCHEMBL28359072

SCHEMBL28359072

CC(C)(C)OC(=O)C(C)(C)c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.51
POLB P06746 1/20 0.51
MAPT P10636 2/20 0.49
LMNA P02545 1/20 0.49
MAPK1 P28482 1/20 0.44
CYP2C19 P33261 1/20 0.44
HSD11B1 P28845 1/20 0.43
CES1 P23141 1/20 0.43
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
GAA P10253 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ACHE P22303 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TSHR P16473 1/20 0.41
NR1D1 P20393 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3530965 0.87 ALDH1A1 (0.51) ALDH1A1POLBMAPTLMNAMAPK1
SCHEMBL429356 0.85 ALDH1A1 (0.65) ALDH1A1POLBMAPTMAPK1CYP2C19
SCHEMBL1646651 0.82 TDP1 (0.52) ALDH1A1POLBLMNAMAPK1HSD11B1
SCHEMBL6680006 0.81 PTPRC (0.54) ALDH1A1POLBMAPTLMNACES1
SCHEMBL395369 0.81 ALDH1A1 (0.56) ALDH1A1POLBMAPTLMNAGAA
SCHEMBL27030901 0.79 MAPT (0.69) ALDH1A1MAPTLMNA
SCHEMBL1647740 0.79 MAPK1 (0.55) ALDH1A1POLBMAPTMAPK1HSD11B1
SCHEMBL6218720 0.78 ALDH1A1 (0.57) ALDH1A1POLBMAPTCYP2C19GAA
SCHEMBL15987513 0.78 CYP2C19 (0.65) ALDH1A1MAPTLMNACYP2C19GAA
SCHEMBL2814601 0.77 MAPT (0.55) ALDH1A1POLBMAPTLMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4619406-A1 TRICYCLIC COMPOUNDS Schrödinger, Inc. (US) 2025-09-24 EP disclosed
WO-2024107393-A1 TRICYCLIC COMPOUNDS SCHRÖDINGER, INC. (US) 2024-05-23 WO disclosed
CN-110818641-B Pyridazine-3-formamide compound, preparation method and application thereof in medicine and pharmacology 北京诺诚健华医药科技有限公司 2022-10-14 CN disclosed
CN-110818641-A Pyridazine-3-formamide compound, preparation method and application thereof in medicine and pharmacology 北京诺诚健华医药科技有限公司 2020-02-21 CN disclosed