SCHEMBL1646834

SCHEMBL1646834

COc1ccccc1NC(=O)CN1CCNCC1

nearest known ligand 0.76

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.76
KMT2A Q03164 7/20 0.68
MEN1 O00255 6/20 0.68
TSHR P16473 3/20 0.65
MAPT P10636 2/20 0.65
LMNA P02545 1/20 0.65
L3MBTL1 Q9Y468 1/20 0.65
RAB9A P51151 1/20 0.65
NPSR1 Q6W5P4 4/20 0.64
CYP2C19 P33261 3/20 0.64
CYP1A2 P05177 2/20 0.64
CYP2C9 P11712 2/20 0.64
SMN1; SMN2 Q16637 4/20 0.63
CYP2D6 P10635 2/20 0.63
USP2 O75604 1/20 0.63
CYP3A4 P08684 1/20 0.63
HTT P42858 1/20 0.63
POLB P06746 1/20 0.63
TP53 P04637 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4559296 0.89 ALDH1A1 (0.60) ALDH1A1KMT2AMEN1TSHRMAPT
SCHEMBL1644836 0.88 ALDH1A1 (0.97) ALDH1A1KMT2AMEN1TSHRMAPT
SCHEMBL29832051 0.87 TDP1 (0.76) ALDH1A1KMT2AMEN1MAPTLMNA
SCHEMBL1646961 0.86 ALDH1A1 (1.00) ALDH1A1KMT2AMEN1TSHRMAPT
SCHEMBL11847704 0.85 ALDH1A1 (0.55) ALDH1A1KMT2AMEN1TSHRLMNA
SCHEMBL1644843 0.85 L3MBTL1 (0.79) ALDH1A1KMT2AMEN1TSHRMAPT
SCHEMBL6169872 0.84 ALDH1A1 (0.76) ALDH1A1KMT2AMEN1TSHRMAPT
SCHEMBL1643927 0.84 ALDH1A1 (0.76) ALDH1A1KMT2AMEN1TSHRMAPT
SCHEMBL1646962 0.84 ALDH1A1 (0.76) ALDH1A1KMT2AMEN1TSHRMAPT
SCHEMBL6175296 0.83 ALDH1A1 (0.74) ALDH1A1KMT2AMEN1TSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4665239-B2 2011-04-06 JP claimed
EP-1071668-A1 5-AMINOINDENO(1,2-C)PYRAZOL-4-ONES AS ANTI-CANCER AND ANTI-PROLIFERATIVE AGENTS Du Pont Pharmaceuticals Company (US) 2001-01-31 EP disclosed
WO-1999054308-A1 5-AMINOINDENO(1,2-C)PYRAZOL-4-ONES AS ANTI-CANCER AND ANTI-PROLIFERATIVE AGENTS DU PONT PHARMACEUTICALS COMPANY (US) 1999-10-28 WO disclosed