SCHEMBL1647433

SCHEMBL1647433

COc1ccc(-c2nn(C3CCCCO3)cc2-c2ccnc(C)c2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.45
TGFBR1 P36897 3/20 0.37
ABL1 P00519 2/20 0.36
BRAF P15056 2/20 0.36
MAPK3 P27361 1/20 0.36
MAPK1 P28482 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CYP3A4 P08684 2/20 0.35
PSEN1 P49768 2/20 0.35
PSEN2 P49810 2/20 0.35
APH1B Q8WW43 2/20 0.35
NCSTN Q92542 2/20 0.35
APH1A Q96BI3 2/20 0.35
PSENEN Q9NZ42 2/20 0.35
KDR P35968 2/20 0.35
MAPK14 Q16539 2/20 0.35
RIPK2 O43353 1/20 0.35
GRM2 Q14416 2/20 0.35
PDE4D Q08499 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1646894 0.89 DYRK1A (0.46) DYRK1AABL1BRAFMAPK3MAPK1
SCHEMBL1646713 0.88 CSNK1D (0.44) TGFBR1ABL1BRAFMAPK3MAPK1
SCHEMBL1646733 0.87 PTGS2 (0.44) BRAFMAPK3MAPK1MEN1KMT2A
SCHEMBL1646295 0.83 BRAF (0.40) ABL1BRAFMEN1KMT2ACYP3A4
SCHEMBL1648278 0.79 AURKB (0.48) BRAFMAPK14
SCHEMBL1645070 0.76 CSNK1D (0.42) ABL1BRAFMAPK3MAPK1MAPK14
SCHEMBL1647734 0.75 CYP1A2 (0.38) ABL1BRAFMAPK1MEN1KMT2A
SCHEMBL1645345 0.75 GRM5 (0.37) BRAFKDRDRD1ALDH1A1HTT
SCHEMBL1646367 0.75 JAK2 (0.41) DYRK1AABL1KDRMAPK14
SCHEMBL1645150 0.74 CSNK1D (0.40) TGFBR1ABL1BRAFMAPK3MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2784070-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2784071-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2784072-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2784073-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2308866-A1 Phenylpyri(mi)dinylpyrazoles and their use as fungicides Bayer CropScience AG (DE) 2011-04-13 EP disclosed