SCHEMBL1647734

SCHEMBL1647734

CCNc1cc(-c2cn(C3CCCCO3)nc2-c2ccc(OC)cc2)ncn1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 5/20 0.38
CYP3A4 P08684 5/20 0.38
TSHR P16473 5/20 0.38
HSD17B10 Q99714 4/20 0.38
USP2 O75604 4/20 0.38
ALDH1A1 P00352 4/20 0.38
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38
HIF1A Q16665 1/20 0.38
FAAH O00519 1/20 0.36
PIK3CA P42336 1/20 0.36
BRAF P15056 1/20 0.36
FLT3 P36888 3/20 0.35
MERTK Q12866 3/20 0.35
KDR P35968 2/20 0.35
FGFR1 P11362 2/20 0.35
AXL P30530 2/20 0.35
AURKA O14965 1/20 0.35
RET P07949 1/20 0.35
SRC P12931 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1645407 0.90 BRAF (0.37) CYP1A2HSD17B10USP2ALDH1A1CASP1
SCHEMBL1645345 0.79 GRM5 (0.37) HSD17B10ALDH1A1BRAFFLT3KDR
SCHEMBL1646295 0.77 BRAF (0.40) CYP1A2CYP3A4TSHRHSD17B10USP2
SCHEMBL1646733 0.76 PTGS2 (0.44) BRAFKDRMAPK1MEN1KMT2A
SCHEMBL1646367 0.76 JAK2 (0.41) KDRFGFR1AURKARETCLK4
SCHEMBL1647433 0.75 DYRK1A (0.45) CYP3A4USP2ALDH1A1BRAFKDR
SCHEMBL1646894 0.75 DYRK1A (0.46) CYP1A2CYP3A4TSHRHSD17B10USP2
SCHEMBL26112883 0.72 EGFR (0.40) CYP1A2CYP3A4TSHRHSD17B10USP2
SCHEMBL1648278 0.72 AURKB (0.48) BRAFAURKACYP2D6
SCHEMBL26115718 0.72 NPC1 (0.41) CYP1A2CYP3A4TSHRHSD17B10USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2784073-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2784070-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2784071-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2784072-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2308866-A1 Phenylpyri(mi)dinylpyrazoles and their use as fungicides Bayer CropScience AG (DE) 2011-04-13 EP disclosed