SCHEMBL16477751

SCHEMBL16477751

Cc1cccc(CN2CCC(N(C)C(=O)COc3nc(C)c(N)c(C)n3)CC2)c1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 2/20 0.43
LTA4H P09960 1/20 0.43
ALDH1A1 P00352 2/20 0.43
HTT P42858 1/20 0.43
DRD4 P21917 3/20 0.42
KCNH2 Q12809 1/20 0.42
DRD2 P14416 2/20 0.42
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
HTR2B P41595 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
FAAH O00519 1/20 0.41
CCR3 P51677 1/20 0.41
KDM4E B2RXH2 1/20 0.41
CHRM2 P08172 1/20 0.40
CHRM3 P20309 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13354219 0.91 MCHR1 (0.44) MCHR1LTA4HALDH1A1KCNH2DRD2
SCHEMBL2850149 0.91 KCNH2 (0.52) MCHR1ALDH1A1DRD4KCNH2DRD2
SCHEMBL13173232 0.90 ALDH1A1 (0.52) MCHR1ALDH1A1DRD4SIGMAR1MEN1
Bromide SCHEMBL2840704 0.90 KCNH2 (0.51) MCHR1ALDH1A1DRD4KCNH2DRD2
Hydrochloric Acid SCHEMBL2841731 0.90 KCNH2 (0.51) MCHR1ALDH1A1DRD4KCNH2DRD2
Hydrochloric Acid SCHEMBL2848182 0.89 ALDH1A1 (0.52) MCHR1ALDH1A1DRD4SIGMAR1MEN1
SCHEMBL2849321 0.89 KCNH2 (0.50) MCHR1ALDH1A1HTTDRD4KCNH2
Maleic Acid SCHEMBL2845354 0.86 SIGMAR1 (0.55) ALDH1A1DRD4KCNH2DRD2HTR2A
SCHEMBL3155541 0.86 KMT2A (0.46) LTA4HALDH1A1DRD4KCNH2SIGMAR1
Fumaric Acid SCHEMBL2845369 0.86 SIGMAR1 (0.55) ALDH1A1DRD4KCNH2DRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2679586-A1 Nitrogen-containing six-membered aromatic ring derivatives and pharmaceutical products containing the same Daiichi Sankyo Company, Limited (JP) 2014-01-01 EP disclosed