SCHEMBL1647835

SCHEMBL1647835

CC(C)=CCn1ncc(-c2ccncc2)c1-c1ccc(F)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.54
PTGS2 P35354 1/20 0.54
MAPK14 Q16539 13/20 0.43
KDR P35968 1/20 0.42
NPC1 O15118 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
NFKB1 P19838 1/20 0.42
RAB9A P51151 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
S1PR1 P21453 1/20 0.41
MAPK13 O15264 4/20 0.40
MAPK12 P53778 4/20 0.40
MAPK11 Q15759 4/20 0.40
CSNK1D P48730 2/20 0.40
MAP4K4 O95819 1/20 0.40
MAPK9 P45984 1/20 0.40
CSNK1A1 P48729 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1645202 0.82 PTGS1 (0.44) PTGS1PTGS2MAPK14KDRNPC1
SCHEMBL6076416 0.81 MAPK14 (0.51) MAPK14KDRNPC1ALDH1A1MAPT
SCHEMBL1647324 0.79 S1PR1 (0.60) MAPK14KDRNPC1ALDH1A1MAPT
SCHEMBL5451477 0.76 MAPK14 (0.47) MAPK14KDRNPC1ALDH1A1MAPT
SCHEMBL6077636 0.75 S1PR1 (0.44) MAPK14KDRNPC1ALDH1A1MAPT
SCHEMBL1645205 0.73 MAPK14 (0.58) PTGS2MAPK14KDRMAPK13MAPK12
SCHEMBL10413532 0.73 MAPK14 (0.59) PTGS2MAPK14ALDH1A1SMN1; SMN2S1PR1
SCHEMBL6078034 0.72 MAPK14 (0.58) MAPK14KDRALDH1A1MAPTS1PR1
SCHEMBL4176192 0.70 PTGS2 (1.00) PTGS1PTGS2
SCHEMBL1554788 0.68 GRIN1 (0.46) MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2784071-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2784070-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2784072-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2784073-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2308866-A1 Phenylpyri(mi)dinylpyrazoles and their use as fungicides Bayer CropScience AG (DE) 2011-04-13 EP disclosed