SCHEMBL16478355

SCHEMBL16478355

CN1Cc2cc(-c3ccc(C(C#N)CNC(=O)C4CCOCC4)cc3)cnc2C1=O

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSC P53634 8/20 0.38
CTSK P43235 4/20 0.38
CYP11B2 P19099 1/20 0.37
WNT1 P04628 2/20 0.37
GSK3B P49841 2/20 0.37
DYRK1A Q13627 2/20 0.37
MAPK1 P28482 4/20 0.34
HDAC6 Q9UBN7 2/20 0.33
HTR1A P08908 1/20 0.33
DRD2 P14416 1/20 0.33
DRD4 P21917 1/20 0.33
ABL1 P00519 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16478224 0.88 CTSC (0.36) CTSCCTSKMAPK1
SCHEMBL289966 0.84 CTSC (0.54) CTSCCTSK
SCHEMBL16478361 0.82 CTSK (0.35) CTSCCTSKCYP11B2
SCHEMBL290330 0.79 CTSC (0.38) CTSCCTSKMAPK1
SCHEMBL16478185 0.79 RET (0.40) CTSCCTSKMAPK1
SCHEMBL16478162 0.77 KCNH2 (0.32) CTSCCTSKCYP11B2
SCHEMBL16478365 0.75 F9 (0.39) CTSCCTSKGSK3BMAPK1
SCHEMBL2890767 0.71 CTSC (0.74) CTSCCTSK
SCHEMBL2890772 0.71 CTSC (0.74) CTSCCTSK
SCHEMBL289965 0.71 CTSC (0.39) CTSCCTSKCYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011154677-A1 SUBSTITUTED N-[1-CYANO-2-(PHENYL)ETHYL] 1-AMINOCYCLOALK-1-YLCARBOXAMIDE COMPOUNDS - 760 ASTRAZENECA AB (SE) 2011-12-15 WO disclosed