SCHEMBL1648049

SCHEMBL1648049

O=C(Nc1cccnc1)c1cccc(OC[C@H]2CCCN2)c1

nearest known ligand 0.63

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.63
MAPK1 P28482 2/20 0.63
ALDH1A1 P00352 3/20 0.57
CHRNB4 P30926 2/20 0.52
CHRNA3 P32297 2/20 0.52
CHRNA1 P02708 1/20 0.52
CHRNG P07510 1/20 0.52
CHRNB1 P11230 1/20 0.52
CHRNB2 P17787 1/20 0.52
CHRNA4 P43681 1/20 0.52
CHRND Q07001 1/20 0.52
KDM4E B2RXH2 1/20 0.52
NR1H4 Q96RI1 1/20 0.51
BRAF P15056 1/20 0.51
GRM5 P41594 1/20 0.49
LMNA P02545 1/20 0.49
HTT P42858 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1648747 0.80 LRRK2 (0.66)
SCHEMBL6917993 0.80 LRRK2 (0.66)
SCHEMBL1648751 0.80 LRRK2 (0.66)
SCHEMBL29039242 0.77 CHRNB4 (0.67) CHRNB4CHRNA3NR1H4
SCHEMBL29039239 0.77 CHRNB4 (0.67) CHRNB4CHRNA3NR1H4
SCHEMBL905236 0.77 CHRNA3 (0.81) CHRNB4CHRNA3CHRNA1CHRNGCHRNB1
SCHEMBL905201 0.77 CHRNA3 (0.81) CHRNB4CHRNA3CHRNA1CHRNGCHRNB1
SCHEMBL3942452 0.77 CHRNA3 (0.81) CHRNB4CHRNA3CHRNA1CHRNGCHRNB1
SCHEMBL26999492 0.77 CHRNB4 (0.63) CHRNB4CHRNA3
SCHEMBL29039262 0.77 CHRNB4 (0.63) CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011038572-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2011-04-07 WO disclosed