SCHEMBL16485759

SCHEMBL16485759

CCC(CC)(NC(=O)OC(C)(C)C)C(=O)N[C@H](C#N)Cc1ccc(-c2ccc(C#N)cc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSC P53634 19/20 0.48
KCNH2 Q12809 5/20 0.48
LTB4R Q15722 1/20 0.46
LTB4R2 Q9NPC1 1/20 0.46
CTSK P43235 4/20 0.46
CTSS P25774 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16485741 0.86 CTSS (0.48) CTSCKCNH2CTSKCTSS
SCHEMBL30195065 0.86 CTSC (0.56) CTSCKCNH2LTB4RLTB4R2CTSK
SCHEMBL20162060 0.86 CTSC (0.56) CTSCKCNH2LTB4RLTB4R2CTSK
SCHEMBL16478084 0.77 CTSC (0.61) CTSCKCNH2LTB4RLTB4R2CTSK
SCHEMBL16478082 0.77 CTSC (0.61) CTSCKCNH2LTB4RLTB4R2CTSK
SCHEMBL16485739 0.77 CTSC (0.58) CTSCKCNH2LTB4RLTB4R2CTSK
SCHEMBL2074657 0.76 CTSC (0.57) CTSCKCNH2CTSKCTSS
SCHEMBL2074655 0.76 CTSC (0.57) CTSCKCNH2CTSKCTSS
SCHEMBL16478098 0.76 CTSC (0.63) CTSCKCNH2LTB4RLTB4R2CTSK
SCHEMBL16478099 0.76 CTSC (0.63) CTSCKCNH2LTB4RLTB4R2CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011154677-A1 SUBSTITUTED N-[1-CYANO-2-(PHENYL)ETHYL] 1-AMINOCYCLOALK-1-YLCARBOXAMIDE COMPOUNDS - 760 ASTRAZENECA AB (SE) 2011-12-15 WO disclosed