Cariporide

Cariporide

SCHEMBL1648723

CC(C)c1ccc(C(=O)N=C(N)N)cc1S(C)(=O)=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 5/20 1.00
SLC9A2 Q9UBY0 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cariporide SCHEMBL31563713 1.00 SLC9A1 (1.00) SLC9A1SLC9A2
Cariporide SCHEMBL8743795 0.99 SLC9A1 (0.97) SLC9A1SLC9A2
Cariporide SCHEMBL611696 0.97 SLC9A1 (1.00) SLC9A1SLC9A2
Hydrochloric Acid SCHEMBL8816755 0.87 SLC9A1 (0.78) SLC9A1SLC9A2
SCHEMBL8573607 0.87 SLC9A1 (0.78) SLC9A1SLC9A2
SCHEMBL8743809 0.87 SLC9A1 (0.76) SLC9A1SLC9A2
Hydrochloric Acid SCHEMBL8743818 0.85 SLC9A1 (0.74) SLC9A1SLC9A2
SCHEMBL7798624 0.85 SLC9A1 (0.74) SLC9A1SLC9A2
SCHEMBL8647605 0.84 SLC9A1 (0.72) SLC9A1SLC9A2
SCHEMBL4355373 0.83 SLC9A1 (0.72) SLC9A1SLC9A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 101 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1146863-B1 LYOPHILISATES WITH IMPROVED RECONSTITUTIBILITY MERCK PATENT GMBH (DE) 2004-05-12 EP claimed
CN-1367689-A Use of sodium-hydrogen exchanger inhibitors for producing medicaments for preventing organ dysfunction and diseases caused by aging and for prolonging life AVENTIS PHARMA GMBH (DE) 2002-09-04 CN claimed
US-6420430-B1 USE OF BENZOYLGUANIDINE DERIVATIVES TO PREVENT AGING DISORDERS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2002-07-16 US claimed
EP-1140056-A2 THE UTILISATION OF INHIBITORS OF THE SODIUM HYDROGEN EXCHANGER FOR PRODUCING A MEDICAMENT FOR PREVENTING ORGAN DYSFUNCTIONS AND DISEASES RELATED TO A PARTICULAR AGE AND FOR PROLONGING LIFE Aventis Pharma Deutschland GmbH (DE) 2001-10-10 EP claimed
WO-2000038661-A2 THE UTILISATION OF INHIBITORS OF THE SODIUM HYDROGEN EXCHANGER FOR PRODUCING A MEDICAMENT FOR PREVENTING ORGAN DYSFUNCTIONS AND DISEASES RELATED TO A PARTICULAR AGE AND FOR PROLONGING LIFE AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-07-06 WO claimed
EP-4709753-A1 SLC4A4/NBCE1 INHIBITORS VIB VZW (BE) 2026-03-18 EP disclosed
US-20250262239-A1 METHOD OF ADMINISTRATION AND TREATMENT DYVE BIOSCIENCES, INC. 2025-08-21 US disclosed
US-12310983-B2 Method of administration and treatment DYVE BIOSCIENCES, INC. (US) 2025-05-27 US disclosed
WO-2024231348-A1 SLC4A4/NBCE1 INHIBITORS VIB VZW (BE) 2024-11-14 WO disclosed
US-12016856-B2 Compounds and methods for inhibiting NHE-mediated antiport in the treatment of disorders associated with fluid retention or salt overload and gastrointestinal tract disorders ARDELYX, INC. (US) 2024-06-25 US disclosed
US-12016856-B2 Compounds and methods for inhibiting NHE-mediated antiport in the treatment of disorders associated with fluid retention or salt overload and gastrointestinal tract disorders ARDELYX, INC. (US) 2024-06-25 US disclosed
EP-4324460-A2 SODIUM BICARBONATE FOR USE IN THE TREATMENT OF GOUT AND RELATED DISORDERS Dyve Biosciences, Inc. (US) 2024-02-21 EP disclosed
US-6844361-B2 Pharmaceutical composition comprising a sodium hydrogen exchange inhibitor and an angiotensin converting enzyme inhibitor AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2005-01-18 US disclosed
WO-2003068212-A1 USE OF SODIUM/HYDROGEN EXCHANGE INHIBITORS FROM THE TREATMENT OF THROMBOTIC AND INFLAMMATORY DISEASES AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2003-08-21 WO disclosed
JP-2002105043-A INTERMEDIATE COMPOUND FOR PRODUCING DIACYL-SUBSTITUTED GUANIDINE HOECHST AG 2002-04-10 JP disclosed
EP-0918515-A2 USE OF INHIBITORS OF THE CELLULAR Na?+ /H?+ EXCHANGER (NHE) FOR PREPARING A MEDICAMENT FOR NORMALIZING SERUM LIPIDS HOECHST AKTIENGESELLSCHAFT (DE) 1999-06-02 EP disclosed
WO-1997046226-A2 USE OF INHIBITORS OF THE CELLULAR Na+/H+ EXCHANGER (NHE) FOR PREPARING A MEDICAMENT FOR NORMALIZING SERUM LIPIDS HOECHST AKTIENGESELLSCHAFT (DE) 1997-12-11 WO disclosed
EP-0589336-B1 Benzoylguanidines, process for their preparation and their use as antiarrhythmic agents HOECHST AG (DE) 1997-01-08 EP disclosed
US-5591754-A Benzoylguanidines, pharmaceutical composition containing them and treatment of arrthythmias therewith HOECHST AKTIENGESELLSCHAFT (DE) 1997-01-07 US disclosed
EP-0589336-A1 Benzoylguanidines, process for their preparation and their use as antiarrhythmic agents HOECHST AKTIENGESELLSCHAFT (DE) 1994-03-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12016856-B2 Compounds and methods for inhibiting NHE-mediated antiport in the treatment of disorders associated with fluid retention or salt overload and gastrointestinal tract disorders SLC10A1, SLC10A2, FABP3 SLC9A1 10/4885SLC9A2 6/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.