SCHEMBL16488478

SCHEMBL16488478

N=C(N)NCCC[C@@H]1NC(=O)CNC(=O)CNC(=O)[C@H](CCC(N)=O)NC(=O)[C@@H]2CCCN2C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CC(=O)O)NC(=O)CNC1=O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.61
ITGAV P06756 1/20 0.61
ITGA2B P08514 1/20 0.61
KLKB1 P03952 4/20 0.57
MC4R P32245 7/20 0.55
MC5R P33032 7/20 0.55
MC3R P41968 7/20 0.55
MC1R Q01726 7/20 0.55
TSLP Q969D9 6/20 0.54
HDAC3 O15379 1/20 0.54
HDAC4 P56524 1/20 0.54
HDAC1 Q13547 1/20 0.54
HDAC7 Q8WUI4 1/20 0.54
HDAC2 Q92769 1/20 0.54
HDAC10 Q969S8 1/20 0.54
HDAC11 Q96DB2 1/20 0.54
HDAC8 Q9BY41 1/20 0.54
HDAC6 Q9UBN7 1/20 0.54
HDAC9 Q9UKV0 1/20 0.54
HDAC5 Q9UQL6 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22193885 0.87 ITGB3 (0.81) ITGB3ITGAVITGA2BKLKB1MC4R
SCHEMBL24433365 0.87 ITGB3 (0.81) ITGB3ITGAVITGA2BKLKB1MC4R
SCHEMBL30866243 0.86 HDAC3 (0.58) ITGB3ITGAVITGA2BHDAC3HDAC4
Eptifibatide SCHEMBL8284422 0.85 ITGB3 (0.82) ITGB3ITGAVITGA2BMC4RMC5R
Eptifibatide SCHEMBL29398425 0.85 ITGB3 (0.82) ITGB3ITGAVITGA2BMC4RMC5R
Eptifibatide SCHEMBL15781 0.85 ITGB3 (0.82) ITGB3ITGAVITGA2BMC4RMC5R
Eptifibatide SCHEMBL571287 0.85 ITGB3 (0.82) ITGB3ITGAVITGA2BMC4RMC5R
SCHEMBL30169340 0.85 HDAC3 (0.59) ITGB3ITGAVITGA2BMC4RMC5R
Eptifibatide SCHEMBL21753462 0.85 ITGB3 (0.81) ITGB3ITGAVITGA2BMC4RMC5R
Eptifibatide SCHEMBL7107217 0.85 ITGB3 (0.81) ITGB3ITGAVITGA2BMC4RMC5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160326217-A1 Methods and Compositions Related to Cyclic Peptide Synthesis NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2016-11-10 US disclosed
EP-1998792-B1 METHODS AND COMPOSITIONS RELATED TO CYCLIC PEPTIDE SYNTHESIS UNIV UTAH RES FOUND (US) 2015-02-18 EP disclosed