SCHEMBL1649443

SCHEMBL1649443

COC(=O)C1=C(C(=O)OC)NC=CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PYGM P11217 1/20 0.52
ALDH1A1 P00352 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
CHRM3 P20309 1/20 0.33
SLC6A3 Q01959 6/20 0.32
TSHR P16473 1/20 0.31
SLC6A2 P23975 2/20 0.31
SLC6A4 P31645 1/20 0.31
CA12 O43570 3/20 0.31
CA1 P00915 3/20 0.31
CA2 P00918 3/20 0.31
CA7 P43166 3/20 0.31
CA9 Q16790 3/20 0.31
CA14 Q9ULX7 3/20 0.31
TDP1 Q9NUW8 1/20 0.31
NPSR1 Q6W5P4 1/20 0.30
NR4A2 P43354 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9671898 0.81 PYGM (0.43) PYGMALDH1A1CHRM3SLC6A3TSHR
SCHEMBL12493386 0.75 TSHR (0.41) ALDH1A1CHRM3SLC6A3TSHRSLC6A2
SCHEMBL14502255 0.71 SMN1; SMN2 (0.40) ALDH1A1SLC6A3TSHRTDP1SMN1; SMN2
SCHEMBL15457433 0.67 LMNA (0.39) ALDH1A1SLC6A3TSHRSLC6A2SLC6A4
SCHEMBL10482141 0.64 CHRM3 (0.41) ALDH1A1CHRM3TSHRCA12CA1
SCHEMBL7718910 0.64 CHRM3 (0.37) CHRM3TSHRCA12CA1CA2
SCHEMBL7324854 0.64 TSHR (0.42) PYGMALDH1A1CYP2C9CYP2C19TSHR
SCHEMBL11755378 0.62 NPSR1 (0.46) SLC6A3TSHRSLC6A2SLC6A4CA12
SCHEMBL5607056 0.62 NPSR1 (0.46) SLC6A3TSHRSLC6A2SLC6A4CA12
SCHEMBL11755388 0.62 NPSR1 (0.46) SLC6A3TSHRSLC6A2SLC6A4CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7927613-B2 Pharmaceutical co-crystal compositions UNIVERSITY OF SOUTH FLORIDA (US) 2011-04-19 US disclosed
US-7790905-B2 Pharmaceutical propylene glycol solvate compositions MCNEIL-PPC, INC. (US) 2010-09-07 US disclosed