SCHEMBL16494512

SCHEMBL16494512

CNC(=O)Oc1c(-c2ccc(Oc3ccc(F)cc3)cc2)oc2cc(N(CCO)S(C)(=O)=O)ccc12

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.37
CYP3A4 P08684 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
PTGS2 P35354 1/20 0.36
MMP2 P08253 2/20 0.36
MMP9 P14780 2/20 0.36
SCN9A Q15858 2/20 0.35
FPR2 P25090 1/20 0.35
EDNRB P24530 2/20 0.35
KCNH2 Q12809 1/20 0.35
CNR2 P34972 2/20 0.34
BCHE P06276 1/20 0.34
CNR1 P21554 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16494271 0.87 CYP3A4 (0.40) CYP3A4CYP2C9CYP2C19PTGS2KCNH2
SCHEMBL3395300 0.86 CYP2C9 (0.47) CYP3A4CYP2C9CYP2C19KCNH2
SCHEMBL16494697 0.86 CYP3A4 (0.38) CYP3A4CYP2C9CYP2C19PTGS2SCN9A
SCHEMBL16494591 0.85 CYP3A4 (0.38) CYP3A4CYP2C9CYP2C19PTGS2
SCHEMBL16494437 0.84 CYP2C9 (0.52) CYP3A4CYP2C9CYP2C19KCNH2
SCHEMBL16502209 0.81 SCN9A (0.41) ESR1PTGS2MMP2MMP9SCN9A
SCHEMBL4758453 0.81 CYP2C9 (0.50) CYP3A4CYP2C9CYP2C19KCNH2
SCHEMBL16494105 0.79 PTGS2 (0.36) CYP3A4CYP2C9CYP2C19PTGS2SCN9A
SCHEMBL16494748 0.79 CYP2C9 (0.51) CYP3A4CYP2C9CYP2C19KCNH2
SCHEMBL16494350 0.79 PTGS2 (0.35) CYP3A4CYP2C9CYP2C19PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245023-B1 HETEROCYCLIC ANTIVIRAL COMPOUNDS HOFFMANN LA ROCHE (CH) 2011-12-28 EP claimed