SCHEMBL16494697

SCHEMBL16494697

CCc1cc2c(OC(=O)NC)c(-c3ccc(Oc4ccc(F)cc4)cc3)oc2cc1N(CCO)S(C)(=O)=O

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
PTGS2 P35354 1/20 0.35
SCN9A Q15858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16494271 0.91 CYP3A4 (0.40) CYP3A4CYP2C9CYP2C19PTGS2
SCHEMBL16494591 0.90 CYP3A4 (0.38) CYP3A4CYP2C9CYP2C19PTGS2
SCHEMBL16494437 0.88 CYP2C9 (0.52) CYP3A4CYP2C9CYP2C19
SCHEMBL3394357 0.87 CYP3A4 (0.50) CYP3A4CYP2C9CYP2C19
SCHEMBL16493980 0.87 CYP3A4 (0.34) CYP3A4CYP2C9CYP2C19
SCHEMBL16494512 0.86 ESR1 (0.37) CYP3A4CYP2C9CYP2C19PTGS2SCN9A
SCHEMBL16494748 0.83 CYP2C9 (0.51) CYP3A4CYP2C9CYP2C19
SCHEMBL16494105 0.83 PTGS2 (0.36) CYP3A4CYP2C9CYP2C19PTGS2SCN9A
SCHEMBL16494427 0.83 CYP3A4 (0.38) CYP3A4CYP2C9CYP2C19PTGS2
SCHEMBL16494350 0.83 PTGS2 (0.35) CYP3A4CYP2C9CYP2C19PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245023-B1 HETEROCYCLIC ANTIVIRAL COMPOUNDS HOFFMANN LA ROCHE (CH) 2011-12-28 EP claimed