SCHEMBL1649565

SCHEMBL1649565

COc1cccc(CNC(=O)c2c[nH]c3cc(-c4cn[nH]c4)ccc23)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PRKACA P17612 4/20 1.00
PRKACG P22612 4/20 1.00
PRKACB P22694 4/20 1.00
ROCK2 O75116 18/20 0.88
ROCK1 Q13464 15/20 0.83

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12779311 0.91 ROCK2 (1.00) PRKACAPRKACGPRKACBROCK2ROCK1
SCHEMBL12779315 0.89 ROCK2 (1.00) PRKACAPRKACGPRKACBROCK2ROCK1
SCHEMBL1649824 0.89 PRKACA (0.80) PRKACAPRKACGPRKACBROCK2ROCK1
SCHEMBL1648117 0.88 ROCK2 (1.00) PRKACAPRKACGPRKACBROCK2ROCK1
SCHEMBL12780132 0.88 ROCK2 (1.00) PRKACAPRKACGPRKACBROCK2ROCK1
SCHEMBL12779975 0.87 PRKACA (0.76) PRKACAPRKACGPRKACBROCK2ROCK1
SCHEMBL1647622 0.86 ROCK2 (1.00) PRKACAPRKACGPRKACBROCK2ROCK1
SCHEMBL15968147 0.84 ROCK2 (1.00) PRKACAPRKACGPRKACBROCK2ROCK1
SCHEMBL18685145 0.84 ROCK2 (0.81) PRKACAPRKACGPRKACBROCK2ROCK1
SCHEMBL1647780 0.84 PRKACA (1.00) PRKACAPRKACGPRKACBROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011050245-A1 BICYCLIC HETEROARYLS AS KINASE INHIBITORS FENG YANGBO (US) 2011-04-28 WO disclosed
WO-2011050245-A1 BICYCLIC HETEROARYLS AS KINASE INHIBITORS FENG YANGBO (US) 2011-04-28 WO disclosed