SCHEMBL1649575

SCHEMBL1649575

COc1cccc(CNC(=O)c2cc3cnc(-c4cn[nH]c4)cc3[nH]2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 18/20 1.00
ROCK1 Q13464 15/20 1.00
PRKACA P17612 3/20 0.80
PRKACG P22612 3/20 0.80
PRKACB P22694 3/20 0.80

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12779554 0.89 ROCK2 (1.00) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL30988400 0.85 ROCK2 (1.00) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL1648814 0.85 ROCK2 (1.00) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL12779532 0.84 ROCK2 (0.73) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL1649574 0.82 ROCK1 (0.78) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL1649824 0.82 PRKACA (0.80) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL12779529 0.79 ROCK2 (0.66) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL3812995 0.78 ROCK2 (0.76) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL2735976 0.76 SRC (0.77) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL1647879 0.76 ROCK1 (1.00) ROCK2ROCK1PRKACAPRKACGPRKACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011050245-A1 BICYCLIC HETEROARYLS AS KINASE INHIBITORS FENG YANGBO (US) 2011-04-28 WO disclosed
WO-2011050245-A1 BICYCLIC HETEROARYLS AS KINASE INHIBITORS FENG YANGBO (US) 2011-04-28 WO disclosed