SCHEMBL16497679

SCHEMBL16497679

CC1=C(C(=O)Nc2cccc(Cl)c2)C(c2ccccc2)NC(=S)N1

nearest known ligand 0.64

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.64
SMN1; SMN2 Q16637 3/20 0.60
KDM4E B2RXH2 3/20 0.60
CYP2C9 P11712 1/20 0.58
CYP2C19 P33261 1/20 0.58
GAA P10253 2/20 0.56
MAPT P10636 2/20 0.56
DHFR P00374 2/20 0.52
GUSB P08236 1/20 0.51
CA1 P00915 1/20 0.51
CA2 P00918 1/20 0.51
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
TSHR P16473 1/20 0.49
L3MBTL1 Q9Y468 2/20 0.49
KMT2A Q03164 2/20 0.49
MEN1 O00255 1/20 0.49
FFAR3 O14843 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16497756 0.94 ALDH1A1 (0.62) ALDH1A1SMN1; SMN2KDM4ECYP2C9CYP2C19
SCHEMBL7694783 0.88 ALDH1A1 (0.72) ALDH1A1SMN1; SMN2KDM4ECYP2C9CYP2C19
SCHEMBL16497690 0.88 TSHR (0.64) ALDH1A1KDM4EGAAMAPTNPC1
SCHEMBL16497693 0.86 ALDH1A1 (0.70) ALDH1A1SMN1; SMN2KDM4ECYP2C9CYP2C19
SCHEMBL16511360 0.85 ALDH1A1 (0.62) ALDH1A1SMN1; SMN2KDM4ECYP2C9CYP2C19
SCHEMBL16511484 0.84 ALDH1A1 (0.63) ALDH1A1SMN1; SMN2KDM4ECYP2C9CYP2C19
SCHEMBL16497713 0.83 ALDH1A1 (0.67) ALDH1A1SMN1; SMN2KDM4ECYP2C9CYP2C19
SCHEMBL16497858 0.82 HTT (0.66) ALDH1A1KDM4EGAAMAPTGUSB
SCHEMBL7689750 0.81 ALDH1A1 (0.70) ALDH1A1SMN1; SMN2KDM4ECYP2C9CYP2C19
SCHEMBL10112932 0.81 ALDH1A1 (0.65) ALDH1A1SMN1; SMN2KDM4ECYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011151701-A1 6 - METHYL - 4 - PHENYL - 5 - ( PHENYL OR CYCLOALKYL) CARBAMOYL - 1,2,3, 4 - TETRAHYDROPYRIMIDIN- 2 - ONE DERIVATIVES AS ANTITUBERCULAR AGENTS COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2011-12-08 WO claimed
WO-2011151701-A1 6 - METHYL - 4 - PHENYL - 5 - ( PHENYL OR CYCLOALKYL) CARBAMOYL - 1,2,3, 4 - TETRAHYDROPYRIMIDIN- 2 - ONE DERIVATIVES AS ANTITUBERCULAR AGENTS COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2011-12-08 WO disclosed
WO-2011151701-A1 6 - METHYL - 4 - PHENYL - 5 - ( PHENYL OR CYCLOALKYL) CARBAMOYL - 1,2,3, 4 - TETRAHYDROPYRIMIDIN- 2 - ONE DERIVATIVES AS ANTITUBERCULAR AGENTS COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2011-12-08 WO disclosed