SCHEMBL16498043

SCHEMBL16498043

CC(C)OCCOc1ccc(-c2ccccc2-c2csc(NC3CC3)n2)cn1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FFAR2 O15552 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
TYR P14679 1/20 0.38
CCNK O75909 4/20 0.37
CDK9 P50750 4/20 0.37
NPY5R Q15761 1/20 0.37
ITGB3 P05106 4/20 0.36
ITGA2B P08514 4/20 0.36
PTGES O14684 4/20 0.36
ENPP2 Q13822 1/20 0.35
FYN P06241 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16498013 0.89 CCNK (0.44) FFAR2NPC1RAB9ATYRCCNK
SCHEMBL16498184 0.85 FFAR2 (0.43) FFAR2NPC1RAB9ATYRCCNK
SCHEMBL16498186 0.85 FFAR2 (0.43) FFAR2NPC1RAB9ATYRCCNK
SCHEMBL1915656 0.84 FFAR2 (0.48) FFAR2NPC1RAB9ATYRCCNK
SCHEMBL16498356 0.77 CCNK (0.45) NPC1RAB9ATYRCCNKCDK9
SCHEMBL1915236 0.76 NPC1 (0.47) FFAR2NPC1RAB9ATYRCCNK
SCHEMBL1915663 0.76 AR (0.43) FFAR2NPC1RAB9ACCNKCDK9
SCHEMBL16498003 0.73 NPC1 (0.46) NPC1RAB9ATYRCCNKCDK9
SCHEMBL16498495 0.72 RAB9A (0.46) NPC1RAB9ATYRCCNKCDK9
SCHEMBL1915580 0.72 CYP19A1 (0.49) FFAR2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011151434-A1 NOVEL COMPOUNDS, PHARMACEUTICAL COMPOSITION AND METHODS FOR USE IN TREATING METABOLIC DISORDERS EUROSCREEN S.A. (BE) 2011-12-08 WO disclosed