SCHEMBL16503580

SCHEMBL16503580

C=C(O)c1ccc2cccc(-c3ccc(CC)cc3C#N)c2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 2/20 0.38
SLC22A12 Q96S37 5/20 0.37
FNTA P49354 1/20 0.35
FNTB P49356 1/20 0.35
PGGT1B P53609 1/20 0.35
CYP1A2 P05177 2/20 0.34
CYP2A6 P11509 1/20 0.34
GRM5 P41594 1/20 0.32
KDM4E B2RXH2 3/20 0.32
ALDH1A1 P00352 2/20 0.32
TSHR P16473 1/20 0.32
CASP1 P29466 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
TDP1 Q9NUW8 2/20 0.31
NPC1 O15118 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
MAPK1 P28482 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7906709 0.82 CA1 (0.41) XDHSLC22A12CYP1A2KDM4ECYP2C9
SCHEMBL25598480 0.77 BCL2 (0.46) XDHGRM5
SCHEMBL7913890 0.71 KDM4E (0.38) SLC22A12CYP1A2KDM4ECYP2C9CYP2C19
SCHEMBL16502459 0.70 XDH (0.44) XDHSLC22A12GRM5
SCHEMBL16502485 0.70 XDH (0.44) XDHSLC22A12
SCHEMBL16509469 0.70 KDM4E (0.51) XDHKDM4E
SCHEMBL16502465 0.70 SLC22A12 (0.46) XDHSLC22A12CYP1A2CYP2C9CYP2C19
SCHEMBL16509499 0.69 NPC1 (0.43) XDHCYP1A2ALDH1A1CYP2C9CYP2C19
SCHEMBL16502483 0.69 PLAU (0.42) XDHKDM4EALDH1A1NPC1MAPT
SCHEMBL16502455 0.69 GRM5 (0.41) XDHGRM5KDM4ENPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2394987-A1 ACYLGUANIDINE DERIVATIVE Astellas Pharma Inc. (JP) 2011-12-14 EP disclosed