SCHEMBL16504285

SCHEMBL16504285

O=C(Cc1ccccc1C(F)(F)I)Nc1cc(Oc2ccc3nc(NC(=O)C4CC4)sc3n2)ccc1F

nearest known ligand 0.64

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RIPK3 Q9Y572 17/20 0.64
RIPK1 Q13546 17/20 0.64
BRAF P15056 3/20 0.64
KDR P35968 2/20 0.54
CHEK1 O14757 1/20 0.51
IKBKB O14920 1/20 0.51
RAF1 P04049 1/20 0.51
PDGFA P04085 1/20 0.51
CDK1 P06493 1/20 0.51
PDGFRB P09619 1/20 0.51
CCNB1 P14635 1/20 0.51
CCNA2 P20248 1/20 0.51
FGFR3 P22607 1/20 0.51
CDK2 P24941 1/20 0.51
GSK3B P49841 1/20 0.51
MAP2K1 Q02750 1/20 0.51
TEK Q02763 1/20 0.51
MAPK14 Q16539 1/20 0.51
AURKB Q96GD4 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2452621 0.94 RIPK1 (0.70) RIPK3RIPK1BRAFKDRCHEK1
SCHEMBL2456245 0.85 BRAF (0.64) RIPK3RIPK1BRAFKDR
SCHEMBL2452470 0.85 BRAF (0.69) RIPK3RIPK1BRAFKDR
SCHEMBL2453065 0.83 BRAF (0.67) RIPK3RIPK1BRAFKDRCHEK1
SCHEMBL2453182 0.83 RIPK1 (0.80) RIPK3RIPK1BRAFKDRCHEK1
SCHEMBL2453162 0.81 BRAF (0.66) RIPK3RIPK1BRAFKDRCHEK1
SCHEMBL2851381 0.81 BRAF (0.77) RIPK3RIPK1BRAFKDRPDGFRB
SCHEMBL2455436 0.78 BRAF (0.64) RIPK3RIPK1BRAFKDR
SCHEMBL2454632 0.78 BRAF (0.70) RIPK3RIPK1BRAFKDR
SCHEMBL2452667 0.78 BRAF (0.65) RIPK3RIPK1BRAFKDRCHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2399921-A1 HETEROCYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2011-12-28 EP disclosed