Phthalimide

Phthalimide

SCHEMBL165345

Br.O=C1NC(=O)c2ccccc21

nearest known ligand 0.94

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Phthalimide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.94
CASP7 P55210 3/20 0.75
CASP3 P42574 2/20 0.75
CASP6 P55212 2/20 0.75
CASP8 Q14790 2/20 0.75
CASP2 P42575 1/20 0.75
PARP1 P09874 4/20 0.56
PDGFRA P16234 1/20 0.56
FER P16591 1/20 0.56
LTK P29376 1/20 0.56
CDK8 P49336 1/20 0.56
ACVR1 Q04771 1/20 0.56
LRRK2 Q5S007 1/20 0.56
DYRK1B Q9Y463 1/20 0.56
MAPK1 P28482 4/20 0.52
LMNA P02545 3/20 0.52
SMN1; SMN2 Q16637 3/20 0.52
HSD17B10 Q99714 1/20 0.52
MAOA P21397 5/20 0.50
MAOB P27338 4/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phthalimide SCHEMBL4322817 1.00 GSK3B (0.94) GSK3BCASP7CASP3CASP6CASP8
Phthalimide SCHEMBL14764095 0.97 GSK3B (0.88) GSK3BCASP7CASP3CASP6CASP8
Phthalimide SCHEMBL10192661 0.97 GSK3B (1.00) GSK3BCASP7CASP3CASP6CASP8
Phthalimide SCHEMBL30125197 0.97 GSK3B (1.00) GSK3BCASP7CASP3CASP6CASP8
Phthalimide SCHEMBL28226707 0.97 GSK3B (1.00) GSK3BCASP7CASP3CASP6CASP8
Phthalimide SCHEMBL7771670 0.97 GSK3B (1.00) GSK3BCASP7CASP3CASP6CASP8
Phthalimide SCHEMBL29366030 0.97 GSK3B (1.00) GSK3BCASP7CASP3CASP6CASP8
Phthalimide SCHEMBL64 0.97 GSK3B (1.00) GSK3BCASP7CASP3CASP6CASP8
Phthalimide SCHEMBL11040503 0.97 GSK3B (1.00) GSK3BCASP7CASP3CASP6CASP8
Phthalimide SCHEMBL5742518 0.94 GSK3B (0.94) GSK3BCASP7CASP3CASP6CASP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 40 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116444476-B Preparation method of polyketone anticancer natural product Naphthospironone A 南开大学 2024-08-09 CN claimed
CN-106336349-B Bromo trifluoromethoxy compound and its synthetic method 南京优氟医药科技有限公司 2019-08-02 CN claimed
CN-109233131-A A kind of flame retardant type high durable ASA co-extrusion materials 浙江宏博新型建材有限公司 2019-01-18 CN claimed
CN-109134460-A A kind of synthetic method of B-carboline class compound 南开大学 2019-01-04 CN claimed
CN-109020814-A A kind of polysubstituted 10- hydroxyl is luxuriant and rich with fragrance and its derivative and its synthetic method 南开大学 2018-12-18 CN claimed
CN-108117645-A The poly- fragrant acid imide manufacturing method of one kind and its process units 梅雪 2018-06-05 CN claimed
CN-106336349-A Bromotrifluoromethoxy compound and synthetic method thereof 南开大学 2017-01-18 CN claimed
CN-101887773-B Insulated cable, component for control system and manufacturing method of component for control system NGK SPARK PLUG CO 2014-08-06 CN claimed
CN-101887773-A Insulated cable, control system are with parts and control system member manufacturing method NGK SPARK PLUG CO 2010-11-17 CN claimed
CN-116444476-B Preparation method of polyketone anticancer natural product Naphthospironone A 南开大学 2024-08-09 CN disclosed
CN-116444476-A Preparation method of polyketone anticancer natural product Naphthospironone A 南开大学 2023-07-18 CN disclosed
CN-106795105-B Novel method for producing azodicarbonamide 杭州海虹精细化工有限公司 2019-11-15 CN disclosed
CN-110446725-A The manufacturing method of polymer, the compound and polymer for causing group containing free radical polymerization DAINICHISEIKA COLOR CHEM 2019-11-12 CN disclosed
CN-110204525-A Novel fluoro unsaturated cyclic carbonic ester and its manufacturing method 大金工业株式会社 2019-09-06 CN disclosed
EP-2611860-A1 EXPANDED POLYOLEFIN CONTAINING POWDERED ACTIVATED CARBON Kaneka Belgium N.V. (BE) 2013-07-10 EP disclosed
US-20130158141-A1 EXPANDED POLYOLEFIN CONTAINING POWDERED ACTIVATED CARBON KANEKA BELGIUM N.V. (BE) 2013-06-20 US disclosed
WO-2012056320-A1 EXPANDED POLYOLEFIN CONTAINING POWDERED ACTIVATED CARBON KANEKA BELGIUM N.V. (BE) 2012-05-03 WO disclosed
WO-2012028953-A1 EXPANDED POLYOLEFIN CONTAINING POWDERED ACTIVATED CARBON KANEKA BELGIUM N.V. (BE) 2012-03-08 WO disclosed
CN-101887773-A Insulated cable, control system are with parts and control system member manufacturing method NGK SPARK PLUG CO 2010-11-17 CN disclosed
US-5468424-A Mixture of powders or particles of antimony oxide and lead stabilizer with plasticizers AMSPEC CHEMICAL CO., INC. (US) 1995-11-21 US disclosed