SCHEMBL165406

SCHEMBL165406

COc1ncc(-c2cc(F)ccc2N2CCN(C(=O)Cn3ccc4cccnc43)CC2)cn1.CS(=O)(=O)C1CCN(c2ncc(-c3cc(F)ccc3N3CCN(C(=O)Cn4cnc5cccnc54)CC3)cn2)CC1

nearest known ligand 0.43

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 20/20 0.43
KCNH2 Q12809 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL115459 0.91 CXCR3 (0.48) CXCR3
SCHEMBL165563 0.91 GRM5 (0.41) CXCR3KCNH2
SCHEMBL3739124 0.85 CXCR3 (0.53) CXCR3KCNH2
SCHEMBL3735661 0.85 CXCR3 (0.46) CXCR3KCNH2
SCHEMBL3726521 0.82 CXCR3 (0.51) CXCR3KCNH2
SCHEMBL163154 0.82 GRM5 (0.43) CXCR3KCNH2
SCHEMBL3736137 0.81 CXCR3 (0.54) CXCR3KCNH2
SCHEMBL165659 0.81 CXCR3 (0.48) CXCR3KCNH2
SCHEMBL3735551 0.81 GRM5 (0.46) CXCR3
SCHEMBL3726519 0.81 CXCR3 (0.55) CXCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2424840-A1 CXCR3 RECEPTOR ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2012-03-07 EP disclosed
WO-2010126811-A1 CXCR3 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-11-04 WO disclosed