SCHEMBL16542017

SCHEMBL16542017

Cc1ccc(Oc2cc(O)ccc2N)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
TEAD4 Q15561 1/20 0.47
ALDH1A1 P00352 5/20 0.46
POLB P06746 1/20 0.46
MAPT P10636 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
ACHE P22303 1/20 0.41
GAA P10253 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
ESR1 P03372 1/20 0.40
ESR2 Q92731 1/20 0.40
CYP3A4 P08684 1/20 0.39
ICAM1 P05362 1/20 0.39
SELE P16581 1/20 0.39
VCAM1 P19320 1/20 0.39
CCNC P24863 1/20 0.39
CDK8 P49336 1/20 0.39
LTA4H P09960 1/20 0.38
ALOX15 P16050 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12474471 0.86 LTA4H (0.57) MEN1KMT2AALDH1A1MAPTTDP1
SCHEMBL10999189 0.85 TEAD4 (0.54) MEN1KMT2ATEAD4ALDH1A1POLB
SCHEMBL5583654 0.83 TEAD4 (0.57) MEN1KMT2ATEAD4ALDH1A1POLB
SCHEMBL17527050 0.83 NR4A1 (0.42) MEN1KMT2AALDH1A1MAPTTDP1
SCHEMBL17527030 0.83 TSHR (0.44) MEN1KMT2AALDH1A1MAPTTDP1
SCHEMBL4867071 0.81 CAMK2A (0.54) ALDH1A1GAACYP3A4LTA4HHSD17B10
SCHEMBL14283765 0.81 MAOB (0.53) MEN1KMT2ATEAD4ALDH1A1POLB
SCHEMBL17506817 0.81 CYP3A4 (0.43) MEN1KMT2AALDH1A1POLBMAPT
SCHEMBL17498442 0.80 CA14 (0.44) MEN1KMT2AALDH1A1POLBMAPT
SCHEMBL9715074 0.79 MEN1 (0.56) MEN1KMT2AALDH1A1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2536726-B1 DIARYL ETHER LINKED PYRROLO [2,1-C][1,4]BENZODIAZEPINE HYBRIDS AND PROCESS FOR THE PREPARATION THEREOF COUNCIL SCIENT IND RES (IN) 2015-03-04 EP disclosed