SCHEMBL16551971

SCHEMBL16551971

COC(=O)c1nc(CNC(=O)OC(C)(C)C)ccc1SC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 3/20 0.43
CA12 O43570 4/20 0.40
CA1 P00915 4/20 0.40
CA2 P00918 4/20 0.40
CA9 Q16790 4/20 0.40
KDM4A O75164 1/20 0.39
HTT P42858 1/20 0.37
ATR Q13535 1/20 0.37
DYRK1A Q13627 1/20 0.36
MAPT P10636 1/20 0.36
RECQL P46063 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
NAMPT P43490 1/20 0.35
POLB P06746 1/20 0.35
MAPK1 P28482 1/20 0.35
ATM Q13315 1/20 0.35
BCHE P06276 1/20 0.34
CACNA1H O95180 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16551972 0.89 KDM4A (0.40) L3MBTL1CA12CA1CA2CA9
SCHEMBL16551911 0.82 CA12 (0.42) L3MBTL1CA12CA1CA2CA9
SCHEMBL16551977 0.82 L3MBTL1 (0.36) L3MBTL1CA12CA1CA2CA9
SCHEMBL16551914 0.80 KDM4A (0.36) L3MBTL1CA12CA1CA2CA9
SCHEMBL16552124 0.80 NPSR1 (0.40) L3MBTL1MAPTRECQLNPSR1POLB
SCHEMBL16552190 0.78 KDM4A (0.39) L3MBTL1KDM4AHTTATRKDM4E
SCHEMBL20833996 0.78 CKS1B (0.32) L3MBTL1CA12CA1CA2CA9
SCHEMBL18099416 0.77 L3MBTL1 (0.53) L3MBTL1MAPTNPSR1KDM4ELMNA
SCHEMBL5270836 0.77 ATR (0.51) L3MBTL1CA12CA1CA2CA9
SCHEMBL16551880 0.77 MAPT (0.39) L3MBTL1HTTMAPTRECQLNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3042913-A1 CYCLIC PEPTIDE COMPOUND, AND PREPARATION METHOD, PHARMACEUTICAL COMPOSITION AND USE THEREOF Hangzhou Guanyu Bio-Medical Co., Ltd (CN) 2016-07-13 EP disclosed
WO-2015027959-A1 CYCLIC PEPTIDE COMPOUND, AND PREPARATION METHOD, PHARMACEUTICAL COMPOSITION AND USE THEREOF 上海冠宇生物医药科技有限公司 (CN) 2015-03-05 WO disclosed