SCHEMBL16552191

SCHEMBL16552191

CSc1ccc(C(=O)O)nc1CNC(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4A O75164 1/20 0.40
HTT P42858 1/20 0.38
POLB P06746 1/20 0.38
MAPK1 P28482 1/20 0.38
ATM Q13315 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
BRD4 O60885 4/20 0.37
MAPKAPK2 P49137 3/20 0.36
IDO1 P14902 1/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
NAMPT P43490 1/20 0.35
GRM2 Q14416 1/20 0.35
PRMT5 O14744 1/20 0.35
WDR77 Q9BQA1 1/20 0.35
BCHE P06276 1/20 0.35
CACNA1H O95180 1/20 0.35
CACNA1B Q00975 1/20 0.35
CACNA1C Q13936 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16552190 0.89 KDM4A (0.39) KDM4AHTTPOLBMAPK1ATM
SCHEMBL16552097 0.84 KDM4A (0.36) KDM4AHTTPOLBMAPK1ATM
SCHEMBL20834068 0.83 SSTR4 (0.33) KDM4AIDO1
SCHEMBL16551996 0.82 KDM4A (0.41) KDM4APOLBMAPK1ATML3MBTL1
SCHEMBL16552171 0.81 KDM4A (0.34) KDM4AHTTPOLBMAPK1ATM
SCHEMBL17922712 0.79 PDE5A (0.38) POLBL3MBTL1
SCHEMBL16551972 0.78 KDM4A (0.40) KDM4AHTTPOLBMAPK1ATM
SCHEMBL20833855 0.77 SDCBP (0.42) KDM4AL3MBTL1
SCHEMBL20833966 0.76 SUCNR1 (0.34) POLB
SCHEMBL16552163 0.75 MAPT (0.33) KDM4APOLBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3042913-A1 CYCLIC PEPTIDE COMPOUND, AND PREPARATION METHOD, PHARMACEUTICAL COMPOSITION AND USE THEREOF Hangzhou Guanyu Bio-Medical Co., Ltd (CN) 2016-07-13 EP disclosed
WO-2015027959-A1 CYCLIC PEPTIDE COMPOUND, AND PREPARATION METHOD, PHARMACEUTICAL COMPOSITION AND USE THEREOF 上海冠宇生物医药科技有限公司 (CN) 2015-03-05 WO disclosed