SCHEMBL1655321

SCHEMBL1655321

CCC(=O)OC1CNCCO1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SSTR4 P31391 2/20 0.38
SLC6A2 P23975 6/20 0.33
SLC6A4 P31645 5/20 0.33
CHRM2 P08172 2/20 0.33
CHRM4 P08173 2/20 0.33
CHRM1 P11229 2/20 0.33
CHRM3 P20309 2/20 0.33
ADRB2 P07550 1/20 0.33
HTR1A P08908 1/20 0.33
HTR2A P28223 1/20 0.33
ADRA1A P35348 1/20 0.33
HTR2B P41595 1/20 0.33
SLC6A3 Q01959 1/20 0.33
ADRA2C P18825 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL17111269 0.98 SSTR4 (0.38) SSTR4SLC6A2SLC6A4CHRM2CHRM4
SCHEMBL27125582 0.87 SSTR4 (0.37) SSTR4SLC6A2SLC6A4ADRB2HTR1A
Hydrochloric Acid SCHEMBL17111215 0.83 NAAA (0.39) SSTR4SLC6A2SLC6A4
SCHEMBL7907555 0.83 SSTR4 (0.35) SSTR4SLC6A2
SCHEMBL9205001 0.83 SSTR4 (0.35) SSTR4SLC6A2
SCHEMBL28311920 0.82 CHRM2 (0.35) CHRM2CHRM4CHRM1CHRM3
SCHEMBL28181787 0.81 SLC6A2 (0.33) SSTR4SLC6A2SLC6A4ADRB2HTR1A
SCHEMBL9207735 0.80 SSTR4 (0.38) SSTR4SLC6A2SLC6A4SLC6A3
SCHEMBL7266735 0.80 ALDH1A1 (0.38) SSTR4SLC6A2SLC6A4ADRB2HTR1A
Hydrochloric Acid SCHEMBL23277053 0.79 SSTR4 (0.37) SSTR4SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE46856-E1 Substituted 2,3-dihydroimidazo[1,2-c]quinazoline derivatives useful for treating hyper-proliferative disorders and diseases associated with angiogenesis BAYER INTELLECTUAL PROPERTY GMBH (DE) 2018-05-22 US disclosed
EP-3122747-A1 DIHYDROPYRIMIDINE COMPOUNDS AND THEIR APPLICATION IN PHARMACEUTICALS Sunshine Lake Pharma Co., Ltd. (CN) 2017-02-01 EP disclosed
EP-2096919-B1 SUBSTITUTED 2,3-DIHYDROIMIDAZO[1,2-C]QUINAZOLINE DERIVATIVES USEFUL FOR TREATING HYPER-PROLIFERATIVE DISORDERS AND DISEASES ASSOCIATED WITH ANGIOGENESIS BAYER IP GMBH (DE) 2016-03-02 EP disclosed
WO-2016015605-A1 COMPOUNDS AS CDK SMALL-MOLECULE INHIBITORS AND USES THEREOF SUNSHINE LAKE PHARMA CO., LTD. (CN) 2016-02-04 WO disclosed
WO-2015144093-A1 DIHYDROPYRIMIDINE COMPOUNDS AND THEIR APPLICATION IN PHARMACEUTICALS SUNSHINE LAKE PHARMA CO., LTD. (CN) 2015-10-01 WO disclosed
CN-101541723-B Hydrofluoroether compounds and processes for their preparation and use 3M INNOVATIVE PROPERTIES CO 2014-11-26 CN disclosed
US-20130261113-A1 SUBSTITUTED 2,3-DIHYDROIMIDAZO[1,2-C]QUINAZOLINE DERIVATIVES USEFUL FOR TREATING HYPER-PROLIFERATIVE DISORDERS AND DISEASES ASSOCIATED WITH ANGIOGENESIS BAYER PHARMACEUTICALS CORPORATION 2013-10-03 US disclosed
US-8466283-B2 Substituted 2,3-dihydroimidazo[1,2-c]quinazoline derivatives useful for treating hyper-proliferative disorders and diseases associated with angiogenesis BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-06-18 US disclosed
CN-101625524-B Photoresist composition and pattern forming method SHINETSU CHEMICAL CO JP 2012-11-28 CN disclosed
CN-102591152-A Resist composition and patterning process SHIN ETSU EHEMICAL CO LTD 2012-07-18 CN disclosed
CN-102520581-A Method for forming photoresist pattern SHINETSU CHEMICAL CO 2012-06-27 CN disclosed
CN-102088956-A Use of proguanil for treating skin/mucosal disorders TOLMAR INC 2011-06-08 CN disclosed
US-20110083984-A1 Substituted 2,3-dihydroimidazo[1,2-c]quinazoline Derivatives Useful for Treating Hyper-Proliferative Disorders and Diseases Associated with Angiogenesis BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2011-04-14 US disclosed
CN-101625524-A Photoresist composition and pattern forming method SHINETSU CHEMICAL CO 2010-01-13 CN disclosed
CN-101541723-A Hydrofluoroether compounds and processes for their preparation and use 3M INNOVATIVE PROPERTIES CO (US) 2009-09-23 CN disclosed
EP-2096919-A1 SUBSTITUTED 2,3-DIHYDROIMIDAZO[1,2-C]QUINAZOLINE DERIVATIVES USEFUL FOR TREATING HYPER-PROLIFERATIVE DISORDERS AND DISEASES ASSOCIATED WITH ANGIOGENESIS Bayer Schering Pharma Aktiengesellschaft (DE) 2009-09-09 EP disclosed
WO-2008070150-A1 SUBSTITUTED 2,3-DIHYDROIMIDAZO[1,2-C]QUINAZOLINE DERIVATIVES USEFUL FOR TREATING HYPER-PROLIFERATIVE DISORDERS AND DISEASES ASSOCIATED WITH ANGIOGENESIS BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2008-06-12 WO disclosed
CN-101087755-A Substituted arylacylthioureas and related compounds; inhibitors of viral replication ACHILLION PHARMACEUTICALS INC (US) 2007-12-12 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130261113-A1 SUBSTITUTED 2,3-DIHYDROIMIDAZO[1,2-C]QUINAZOLINE DERIVATIVES USEFUL FOR TREATING HYPER-PROLIFERATIVE DISORDERS AND DISEASES ASSOCIATED WITH ANGIOGENESIS PIK3CA, PIK3CD, PIK3CB SSTR4 4049/4885SLC6A2 3678/4885SLC6A4 4191/4885
US-20110083984-A1 Substituted 2,3-dihydroimidazo[1,2-c]quinazoline Derivatives Useful for Treating Hyper-Proliferative Disorders and Diseases Associated with Angiogenesis PIK3CA, PIK3CD, PIK3CB SSTR4 4049/4885SLC6A2 3678/4885SLC6A4 4191/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.