SCHEMBL16557013

SCHEMBL16557013

OCOCc1ccc2cc(N(c3ccc4nc(COCO)ccc4c3)c3ccc4nc(COCO)ccc4c3)ccc2n1

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 5/20 0.37
CYSLTR1 Q9Y271 4/20 0.37
CYSLTR2 Q9NS75 1/20 0.35
PDE10A Q9Y233 7/20 0.34
ALOX5 P09917 2/20 0.33
ESR1 P03372 1/20 0.33
ESR2 Q92731 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16557000 0.93 PDE10A (0.34) GPBAR1CYSLTR1PDE10AALOX5
SCHEMBL16557009 0.85 TERT (0.35) GPBAR1CYSLTR1CYSLTR2PDE10AALOX5
SCHEMBL14930063 0.84 CYP1A2 (0.40) GPBAR1CYSLTR1PDE10A
SCHEMBL12516193 0.81 CCR1 (0.47) GPBAR1CYSLTR1PDE10A
SCHEMBL12517318 0.77 PDE10A (0.35) GPBAR1CYSLTR1CYSLTR2PDE10AALOX5
SCHEMBL14925219 0.77 PDE10A (0.40) GPBAR1CYSLTR1CYSLTR2PDE10AALOX5
SCHEMBL16557004 0.76 PDE10A (0.33) PDE10A
SCHEMBL2223356 0.74 PDE10A (0.33) GPBAR1CYSLTR1CYSLTR2PDE10A
SCHEMBL14925246 0.73 PDE10A (0.37) GPBAR1CYSLTR1CYSLTR2PDE10AALOX5
SCHEMBL12517340 0.72 CCR1 (0.48) GPBAR1CYSLTR1PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2523937-B1 Multiphoton activable quinoline derivatives, their preparation and their uses CENTRE NAT RECH SCIENT (FR) 2015-03-11 EP disclosed