SCHEMBL1656247

SCHEMBL1656247

C=CCCN(CC[C@H](NC(=O)OC(C)(C)C)C(=O)O)S(=O)(=O)c1ccccc1[N+](=O)[O-].COC(=O)[C@H](CCNCl)C(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.37
TSHR P16473 1/20 0.37
KMT2A Q03164 1/20 0.35
BCL2 P10415 3/20 0.35
GSTP1 P09211 1/20 0.34
GSTM2 P28161 1/20 0.34
NRP1 O14786 1/20 0.34
MCL1 Q07820 1/20 0.34
NPSR1 Q6W5P4 1/20 0.33
PPARA Q07869 2/20 0.33
PPARG P37231 1/20 0.33
JAK3 P52333 1/20 0.32
BTK Q06187 1/20 0.32
CTSK P43235 1/20 0.32
MMP13 P45452 1/20 0.32
P4HB P07237 1/20 0.32
TGM2 P21980 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1052024 0.89 ALDH1A1 (0.41) ALDH1A1TSHRKMT2ABCL2MCL1
SCHEMBL1052027 0.89 ALDH1A1 (0.41) ALDH1A1TSHRKMT2ABCL2MCL1
SCHEMBL1645136 0.87 KMT2A (0.42) ALDH1A1KMT2ABCL2GSTP1GSTM2
SCHEMBL1645137 0.87 KMT2A (0.42) ALDH1A1KMT2ABCL2GSTP1GSTM2
SCHEMBL1644288 0.86 KMT2A (0.44) ALDH1A1KMT2ANPSR1MMP13
SCHEMBL1644292 0.86 KMT2A (0.44) ALDH1A1KMT2ANPSR1MMP13
SCHEMBL12770375 0.84 BCL2 (0.39) KMT2ABCL2MCL1CTSKMMP13
SCHEMBL13059502 0.79 CTSK (0.46) ALDH1A1TSHRPPARAPPARGCTSK
SCHEMBL2235961 0.78 ALDH1A1 (0.39) ALDH1A1TSHRKMT2ABCL2MCL1
SCHEMBL3058638 0.78 ALDH1A1 (0.39) ALDH1A1TSHRKMT2ABCL2MCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2305695-A2 Macrocyclic inhibitors of Hepatitis C virus replication Intermune, Inc. (US) 2011-04-06 EP disclosed
EP-2305697-A2 Macrocyclic inhibitors of Hepatitis C virus replication Intermune, Inc. (US) 2011-04-06 EP disclosed
EP-2305698-A2 Macrocyclic inhibitors of Hepatitis C virus replication Intermune, Inc. (US) 2011-04-06 EP disclosed