SCHEMBL16564597

SCHEMBL16564597

COc1cc(F)ccc1-c1ccnc(Nc2cccc(NS(C)(=O)=O)c2)n1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 17/20 0.63
GSK3A P49840 3/20 0.63
GSK3B P49841 2/20 0.63
CDK5 Q00535 2/20 0.63
MAP4K4 O95819 2/20 0.63
AURKA O14965 1/20 0.63
ABL1 P00519 1/20 0.63
LCK P06239 1/20 0.63
MET P08581 1/20 0.63
PDGFRB P09619 1/20 0.63
FGFR1 P11362 1/20 0.63
FLT1 P17948 1/20 0.63
KDR P35968 1/20 0.63
FLT3 P36888 1/20 0.63
MAPK8 P45983 1/20 0.63
MAPK9 P45984 1/20 0.63
ACVR1 Q04771 1/20 0.63
MST1R Q04912 1/20 0.63
TYRO3 Q06418 1/20 0.63
NTRK2 Q16620 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16564577 0.90 CDK9 (0.77) CDK9GSK3AGSK3BCDK5MAP4K4
Hydrochloric Acid SCHEMBL17257732 0.84 CDK9 (0.77) CDK9GSK3AGSK3BCDK5MAP4K4
SCHEMBL3004001 0.83 CDK9 (0.75) CDK9GSK3AGSK3BCDK5MAP4K4
SCHEMBL12487249 0.81 CDK9 (0.57) CDK9GSK3AGSK3BCDK5MAP4K4
SCHEMBL8516163 0.81 CDK9 (0.81) CDK9GSK3ACDK5MAP4K4LRRK2
SCHEMBL16564576 0.81 CDK9 (0.61) CDK9GSK3AGSK3BCDK5MAP4K4
SCHEMBL14874685 0.80 CDK9 (0.68) CDK9GSK3AGSK3BCDK5MAP4K4
Trifluoroacetic Acid SCHEMBL17257723 0.79 CDK9 (0.68) CDK9GSK3AGSK3BCDK5MAP4K4
SCHEMBL14161111 0.77 CDK9 (1.00) CDK9GSK3AGSK3BCDK5MAP4K4
SCHEMBL15720507 0.75 CDK9 (0.72) CDK9GSK3AGSK3BCDK5CCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2137163-B1 INHIBITORS OF PROTEIN KINASES ASTRAZENECA AB (SE) 2015-03-18 EP claimed