SCHEMBL8516163

SCHEMBL8516163

COc1cc(F)ccc1-c1cc(Nc2cccc(NS(C)(=O)=O)c2)ncn1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 14/20 0.81
CCNT1 O60563 10/20 0.81
MAP4K4 O95819 2/20 0.81
CDK1 P06493 2/20 0.81
CDK4 P11802 2/20 0.81
CCNB1 P14635 2/20 0.81
CCND1 P24385 2/20 0.81
ABL2 P42684 2/20 0.81
GSK3A P49840 2/20 0.81
CDK7 P50613 2/20 0.81
CCNH P51946 2/20 0.81
MNAT1 P51948 2/20 0.81
CYP1A2 P05177 3/20 0.58
CYP2C19 P33261 3/20 0.58
HSD17B10 Q99714 2/20 0.58
USP2 O75604 2/20 0.58
CYP2D6 P10635 2/20 0.58
CLK4 Q9HAZ1 2/20 0.58
ALDH1A1 P00352 1/20 0.58
LMNA P02545 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4096813 0.88 CDK9 (0.69) CDK9CCNT1MAP4K4CDK1CDK4
SCHEMBL2030393 0.85 CDK9 (0.63) CDK9CCNT1MAP4K4CDK1CDK4
SCHEMBL8514160 0.85 CDK9 (0.84) CDK9CCNT1MAP4K4CDK1CDK4
SCHEMBL8515978 0.84 CDK9 (0.66) CDK9CCNT1MAP4K4CDK1CDK4
SCHEMBL12487249 0.84 CDK9 (0.57) CDK9CCNT1MAP4K4CDK1CDK4
SCHEMBL4426442 0.82 CDK9 (0.82) CDK9CCNT1MAP4K4CDK1CDK4
SCHEMBL8516573 0.82 CYP1A2 (0.69) CDK9CCNT1MAP4K4CDK1CDK4
SCHEMBL8515811 0.81 CDK9 (0.80) CDK9CCNT1MAP4K4CDK1CDK4
SCHEMBL16564597 0.81 CDK9 (0.63) CDK9CCNT1MAP4K4CDK1CDK4
SCHEMBL8516178 0.81 CDK9 (0.79) CDK9CCNT1MAP4K4CDK1CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2137166-B1 4, 6-DISUBSTITUTED AMINOPYRIMIDINE DERIVATIVES AS INHIBITORS OF PROTEIN KINASES INGENIUM PHARMACEUTICALS GMBH (DE) 2012-05-30 EP claimed