Esculetin

Esculetin

SCHEMBL165749

O=c1ccc2cc(O)c(O)cc2o1.OC[C@H]1O[C@@H](O)[C@H](O)[C@@H](O)[C@@H]1O

nearest known ligand 0.69

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.69
HPGD P15428 7/20 0.69
KDM4E B2RXH2 6/20 0.69
CASP1 P29466 6/20 0.69
CASP7 P55210 6/20 0.69
HSD17B10 Q99714 6/20 0.69
GAA P10253 5/20 0.69
GLA P06280 4/20 0.69
MEN1 O00255 3/20 0.69
KMT2A Q03164 3/20 0.69
AMY1A P0DUB6 2/20 0.69
CYP2C19 P33261 1/20 0.69
STAT6 P42226 1/20 0.69
ERAP1 Q9NZ08 5/20 0.67
CA9 Q16790 7/20 0.60
CA12 O43570 5/20 0.60
AKR1B1 P15121 3/20 0.60
MCL1 Q07820 3/20 0.60
ACHE P22303 2/20 0.60
CYP1A2 P05177 2/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Esculetin SCHEMBL1707171 1.00 ALDH1A1 (0.69) ALDH1A1HPGDKDM4ECASP1CASP7
Esculin SCHEMBL8155952 0.85 ALDH1A1 (0.96) ALDH1A1HPGDKDM4ECASP1CASP7
SCHEMBL11111897 0.84 ALDH1A1 (0.65) ALDH1A1HPGDKDM4ECASP1CASP7
SCHEMBL13784420 0.83 ALDH1A1 (0.93) ALDH1A1HPGDKDM4ECASP1CASP7
SCHEMBL1536006 0.83 ALDH1A1 (0.93) ALDH1A1HPGDKDM4ECASP1CASP7
SCHEMBL7762578 0.83 ALDH1A1 (0.93) ALDH1A1HPGDKDM4ECASP1CASP7
SCHEMBL29398048 0.83 ALDH1A1 (0.93) ALDH1A1HPGDKDM4ECASP1CASP7
Esculin SCHEMBL13096298 0.82 ALDH1A1 (1.00) ALDH1A1HPGDKDM4ECASP1CASP7
Esculin SCHEMBL2893 0.82 ALDH1A1 (1.00) ALDH1A1HPGDKDM4ECASP1CASP7
Esculin SCHEMBL8035285 0.82 ALDH1A1 (1.00) ALDH1A1HPGDKDM4ECASP1CASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611903-A1 USE OF A BETA-GLUCOSIDASE ACTIVATOR FOR DETECTING AND/OR IDENTIFYING C. DIFFICILE Biomérieux (FR) 2013-07-10 EP claimed
WO-2012028816-A1 USE OF A BETA-GLUCOSIDASE ACTIVATOR FOR DETECTING AND/OR IDENTIFYING C. DIFFICILE bioMérieux (FR) 2012-03-08 WO claimed
EP-2611903-B1 USE OF A BETA-GLUCOSIDASE ACTIVATOR FOR DETECTING AND/OR IDENTIFYING C. DIFFICILE BIOMERIEUX SA (FR) 2016-10-05 EP disclosed
EP-2611903-A1 USE OF A BETA-GLUCOSIDASE ACTIVATOR FOR DETECTING AND/OR IDENTIFYING C. DIFFICILE Biomérieux (FR) 2013-07-10 EP disclosed
WO-2012028816-A1 USE OF A BETA-GLUCOSIDASE ACTIVATOR FOR DETECTING AND/OR IDENTIFYING C. DIFFICILE bioMérieux (FR) 2012-03-08 WO disclosed