SCHEMBL16579802

SCHEMBL16579802

Nc1nc(CCCCc2c[nH]c(N)n2)c[nH]1

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.33
NOS2 P35228 3/20 0.32
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
PDPK1 O15530 2/20 0.31
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1518158 0.90 HRH3 (0.39) PDPK1
SCHEMBL474833 0.90 KCNH2 (0.46) BACE1NOS2PDPK1KCNH2
SCHEMBL1518260 0.89 HRH3 (0.38) PDPK1
SCHEMBL18794910 0.88 KCNH2 (0.48) BACE1NOS2PDPK1KCNH2
SCHEMBL8521631 0.88 KCNH2 (0.48) BACE1NOS2PDPK1KCNH2
Hydrochloric Acid SCHEMBL1518237 0.87 HRH3 (0.37) PDPK1
SCHEMBL12595083 0.85 MIF (0.35) PDPK1
SCHEMBL12598559 0.84 MPO (0.38) BACE1
SCHEMBL365305 0.84
Trifluoroacetic Acid SCHEMBL16566441 0.84 HRH4 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9962383-B2 Compounds, compositions and methods of agelastatin alkaloids MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2018-05-08 US disclosed
US-20170143708-A1 COMPOUNDS, COMPOSITIONS AND METHODS OF AGELASTATIN ALKALOIDS MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2017-05-25 US disclosed
US-9434736-B2 Compounds, compositions and methods of agelastatin alkaloids MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2016-09-06 US disclosed
US-20150080405-A1 COMPOUNDS, COMPOSITIONS AND METHODS OF AGELASTATIN ALKALOIDS MASSACHUSETTS INSTITUTE OF TECHNOLOGY 2015-03-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170143708-A1 COMPOUNDS, COMPOSITIONS AND METHODS OF AGELASTATIN ALKALOIDS DIMT1, CIAPIN1, INMT BACE1 1560/4885NOS2 1128/4885NOS3 804/4885
US-20150080405-A1 COMPOUNDS, COMPOSITIONS AND METHODS OF AGELASTATIN ALKALOIDS DIMT1, CIAPIN1, INMT BACE1 1560/4885NOS2 1128/4885NOS3 804/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.